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6UDX

X-ray co-crystal structure of compound 7 with Mcl-1

Functional Information from GO Data
ChainGOidnamespacecontents
A0042981biological_processregulation of apoptotic process
B0042981biological_processregulation of apoptotic process
Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue Q57 A 401
ChainResidue
APHE228
AHOH563
AHOH612
AHOH614
AVAL249
AMET250
AARG263
ATHR266
ALEU267
APHE270
ALEU290
AHOH518

site_idAC2
Number of Residues12
Detailsbinding site for residue Q57 B 401
ChainResidue
BPHE228
BVAL249
BMET250
BVAL253
BARG263
BLEU267
BPHE270
BLEU290
BHOH553
BHOH557
BHOH559
BHOH600

Functional Information from PROSITE/UniProt
site_idPS01080
Number of Residues20
DetailsBH1 Apoptosis regulator, Bcl-2 family BH1 motif signature. VFsDGvtNWGRIVTLIsFGA
ChainResidueDetails
AVAL253-ALA272

site_idPS01258
Number of Residues12
DetailsBH2 Apoptosis regulator, Bcl-2 family BH2 motif signature. WLvkqRGWDgFV
ChainResidueDetails
ATRP305-VAL316

site_idPS01259
Number of Residues15
DetailsBH3 Apoptosis regulator, Bcl-2 family BH3 motif signature. AletLRrVGDGVQRN
ChainResidueDetails
AALA209-ASN223

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues28
DetailsMotif: {"description":"BH3"}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues40
DetailsMotif: {"description":"BH1"}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues30
DetailsMotif: {"description":"BH2"}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues6
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin)"}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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