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6U72

BRD4-BD1 in complex with the cyclic peptide 3.1_2_AcK5toA

Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for Ligand residues ALY C 12 through GLN C 13 bound to THR C 11
ChainResidue
APHE83
CHOH201
CHOH202
CHOH203
CHOH204
AVAL87
ALEU94
AASN140
AASP144
AASP145
CTHR11
CCYS14
CNH2101

site_idAC2
Number of Residues6
Detailsbinding site for Di-peptide ACE C 0 and TRP C 1
ChainResidue
ALYS141
CLYS2
CTRP9
CARG10
CTHR11
CCYS14

site_idAC3
Number of Residues6
Detailsbinding site for Di-peptide ACE C 0 and CYS C 14
ChainResidue
CTRP1
CARG10
CTHR11
CALY12
CGLN13
CNH2101

site_idAC4
Number of Residues7
Detailsbinding site for Di-peptide GLY C 6 and ALY C 7
ChainResidue
AILE100
BTRP81
CTHR3
CILE4
CALA5
CTHR8
CTRP9

site_idAC5
Number of Residues8
Detailsbinding site for Di-peptide ALY C 7 and THR C 8
ChainResidue
AILE100
BTRP81
CLYS2
CTHR3
CILE4
CALA5
CGLY6
CTRP9

site_idAC6
Number of Residues6
Detailsbinding site for Di-peptide NH2 C 101 and CYS C 14
ChainResidue
CACE0
CTRP1
CARG10
CTHR11
CALY12
CGLN13

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues106
DetailsDomain: {"description":"Bromo 1","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues2
DetailsSite: {"description":"Acetylated histone binding","evidences":[{"source":"PubMed","id":"22464331","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues4
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2)","evidences":[{"source":"PubMed","id":"28112733","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

239492

PDB entries from 2025-07-30

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