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6U63

Mcl-1 bound to compound 17

Functional Information from GO Data
ChainGOidnamespacecontents
A0042981biological_processregulation of apoptotic process
B0042981biological_processregulation of apoptotic process
C0042981biological_processregulation of apoptotic process
D0042981biological_processregulation of apoptotic process
Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue Q0D A 401
ChainResidue
AHIS224
AQ0D402
CTHR226
CALA227
CQ0D500
AMET231
AMET250
AVAL253
APHE254
AARG263
ATHR266
ALEU267
APHE270

site_idAC2
Number of Residues7
Detailsbinding site for residue Q0D A 402
ChainResidue
ALYS234
ALYS308
AQ0D401
BQ0D402
CLYS234
CHIS252
CQ0D500

site_idAC3
Number of Residues12
Detailsbinding site for residue Q0D B 401
ChainResidue
BMET231
BMET250
BVAL253
BPHE254
BARG263
BTHR266
BLEU267
BQ0D402
DTHR226
DALA227
DGLY230
DQ0D500

site_idAC4
Number of Residues4
Detailsbinding site for residue Q0D B 402
ChainResidue
AQ0D402
BHIS252
BQ0D401
CLYS234

site_idAC5
Number of Residues10
Detailsbinding site for residue Q0D C 500
ChainResidue
AALA227
AGLY230
AQ0D401
AQ0D402
CMET231
CVAL253
CPHE254
CARG263
CTHR266
CPHE270

site_idAC6
Number of Residues15
Detailsbinding site for residue Q0D D 500
ChainResidue
BTHR226
BALA227
BGLY230
BMET231
BQ0D401
DMET231
DLEU235
DVAL249
DMET250
DVAL253
DPHE254
DARG263
DTHR266
DLEU267
DPHE270

Functional Information from PROSITE/UniProt
site_idPS01080
Number of Residues20
DetailsBH1 Apoptosis regulator, Bcl-2 family BH1 motif signature. VFsDGvtNWGRIVTLIsFGA
ChainResidueDetails
AVAL253-ALA272

site_idPS01258
Number of Residues12
DetailsBH2 Apoptosis regulator, Bcl-2 family BH2 motif signature. WLvkqRGWDgFV
ChainResidueDetails
ATRP305-VAL316

site_idPS01259
Number of Residues15
DetailsBH3 Apoptosis regulator, Bcl-2 family BH3 motif signature. AletLRrVGDGVQRN
ChainResidueDetails
AALA209-ASN223

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues12
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin)
ChainResidueDetails
CLYS197
DLYS194
DLYS197
ALYS194
ALYS197
BLYS194
BLYS197
CLYS194

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PDB entries from 2024-06-12

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