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6TXA

Crystal structure of tetrameric human D137N-SAMHD1 (residues 109-626) with XTP, dGMPNPP and Mg

Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue FE A 701
ChainResidue
AARG164
AHIS167
AHIS206
AASP207
AASP311
AXG4705

site_idAC2
Number of Residues3
Detailsbinding site for residue MG A 702
ChainResidue
AASP207
AHIS233
AXG4705

site_idAC3
Number of Residues2
Detailsbinding site for residue MG A 703
ChainResidue
AASP309
AXG4705

site_idAC4
Number of Residues2
Detailsbinding site for residue MG A 704
ChainResidue
ACZF706
CXG4701

site_idAC5
Number of Residues18
Detailsbinding site for residue XG4 A 705
ChainResidue
AGLN149
ALEU150
AARG164
AHIS167
AASP207
AHIS210
AHIS215
AHIS233
AASP311
ALYS312
ATYR315
AASP319
AARG366
ATYR374
AGLN375
AFE701
AMG702
AMG703

site_idAC6
Number of Residues14
Detailsbinding site for residue CZF A 706
ChainResidue
ALYS116
AVAL117
AILE118
AASN137
AGLN142
AARG145
APHE165
AMG704
BTYR155
BVAL156
BVAL378
BARG451
CLYS523
CXG4701

site_idAC7
Number of Residues4
Detailsbinding site for residue SO4 A 707
ChainResidue
AARG305
AARG348
AHIS517
AARG531

site_idAC8
Number of Residues17
Detailsbinding site for residue XG4 A 708
ChainResidue
AASP330
AARG333
AARG352
ALYS354
AASN358
ALYS523
CVAL117
CASN119
CMG705
CCZF707
DVAL156
DPHE157
DGLY324
DILE325
DARG372
DHIS376
DLYS377

site_idAC9
Number of Residues7
Detailsbinding site for residue FE B 701
ChainResidue
BARG164
BHIS167
BHIS206
BASP207
BASP311
BMG702
BXG4705

site_idAD1
Number of Residues5
Detailsbinding site for residue MG B 702
ChainResidue
BHIS206
BASP207
BHIS233
BFE701
BXG4705

site_idAD2
Number of Residues3
Detailsbinding site for residue MG B 703
ChainResidue
BASP309
BLYS312
BXG4705

site_idAD3
Number of Residues2
Detailsbinding site for residue MG B 704
ChainResidue
BCZF706
DXG4701

site_idAD4
Number of Residues19
Detailsbinding site for residue XG4 B 705
ChainResidue
BFE701
BMG702
BMG703
BGLN149
BLEU150
BARG164
BHIS167
BASP207
BHIS210
BHIS215
BHIS233
BASP311
BLYS312
BTYR315
BASP319
BARG366
BHIS370
BTYR374
BGLN375

site_idAD5
Number of Residues14
Detailsbinding site for residue CZF B 706
ChainResidue
ATYR155
AVAL156
AVAL378
AARG451
BLYS116
BVAL117
BILE118
BASN137
BGLN142
BARG145
BPHE165
BMG704
DLYS523
DXG4701

site_idAD6
Number of Residues4
Detailsbinding site for residue SO4 B 707
ChainResidue
BARG305
BARG348
BHIS517
BARG531

site_idAD7
Number of Residues19
Detailsbinding site for residue XG4 B 708
ChainResidue
BASP330
BARG333
BARG352
BLYS354
BASN358
BLYS523
CVAL156
CPHE157
CGLY324
CILE325
CARG372
CHIS376
CLYS377
CCZF709
DVAL117
DILE118
DASN119
DHIS125
DMG705

site_idAD8
Number of Residues14
Detailsbinding site for residue XG4 C 701
ChainResidue
AVAL117
AASN119
AMG704
ACZF706
BVAL156
BPHE157
BARG372
BHIS376
BLYS377
CARG333
CARG352
CLYS354
CASN358
CLYS523

site_idAD9
Number of Residues7
Detailsbinding site for residue FE C 702
ChainResidue
CARG164
CHIS167
CHIS206
CASP207
CASP311
CMG703
CXG4706

site_idAE1
Number of Residues5
Detailsbinding site for residue MG C 703
ChainResidue
CHIS206
CASP207
CHIS233
CFE702
CXG4706

site_idAE2
Number of Residues3
Detailsbinding site for residue MG C 704
ChainResidue
CASP309
CLYS312
CXG4706

site_idAE3
Number of Residues2
Detailsbinding site for residue MG C 705
ChainResidue
AXG4708
CCZF707

site_idAE4
Number of Residues19
Detailsbinding site for residue XG4 C 706
ChainResidue
CGLN149
CLEU150
CARG164
CHIS167
CASP207
CHIS210
CHIS215
CHIS233
CASP311
CLYS312
CTYR315
CASP319
CARG366
CHIS370
CTYR374
CGLN375
CFE702
CMG703
CMG704

site_idAE5
Number of Residues14
Detailsbinding site for residue CZF C 707
ChainResidue
ALYS523
AXG4708
CLYS116
CVAL117
CILE118
CASN137
CGLN142
CARG145
CPHE165
CMG705
DTYR155
DVAL156
DVAL378
DARG451

site_idAE6
Number of Residues4
Detailsbinding site for residue SO4 C 708
ChainResidue
CARG305
CARG348
CHIS517
CARG531

site_idAE7
Number of Residues14
Detailsbinding site for residue CZF C 709
ChainResidue
BLYS523
BXG4708
CTYR155
CVAL156
CVAL378
CARG451
DLYS116
DVAL117
DILE118
DASN137
DGLN142
DARG145
DPHE165
DMG705

site_idAE8
Number of Residues17
Detailsbinding site for residue XG4 D 701
ChainResidue
AVAL156
APHE157
AGLY324
AARG372
AHIS376
ALYS377
BVAL117
BASN119
BHIS125
BMG704
BCZF706
DASP330
DARG333
DARG352
DLYS354
DASN358
DLYS523

site_idAE9
Number of Residues7
Detailsbinding site for residue FE D 702
ChainResidue
DARG164
DHIS167
DHIS206
DASP207
DASP311
DMG703
DXG4706

site_idAF1
Number of Residues5
Detailsbinding site for residue MG D 703
ChainResidue
DHIS206
DASP207
DHIS233
DFE702
DXG4706

site_idAF2
Number of Residues2
Detailsbinding site for residue MG D 704
ChainResidue
DASP309
DXG4706

site_idAF3
Number of Residues2
Detailsbinding site for residue MG D 705
ChainResidue
BXG4708
CCZF709

site_idAF4
Number of Residues18
Detailsbinding site for residue XG4 D 706
ChainResidue
DGLN149
DLEU150
DARG164
DHIS167
DASP207
DHIS215
DHIS233
DASP311
DLYS312
DTYR315
DASP319
DARG366
DHIS370
DTYR374
DGLN375
DFE702
DMG703
DMG704

site_idAF5
Number of Residues4
Detailsbinding site for residue SO4 D 707
ChainResidue
DARG305
DARG348
DHIS517
DARG531

site_idAF6
Number of Residues7
Detailsbinding site for residue FE E 701
ChainResidue
EARG164
EHIS167
EHIS206
EASP207
EASP311
EMG702
EXG4705

site_idAF7
Number of Residues5
Detailsbinding site for residue MG E 702
ChainResidue
EHIS206
EASP207
EHIS233
EFE701
EXG4705

site_idAF8
Number of Residues3
Detailsbinding site for residue MG E 703
ChainResidue
EASP309
ELYS312
EXG4705

site_idAF9
Number of Residues2
Detailsbinding site for residue MG E 704
ChainResidue
ECZF706
GXG4701

site_idAG1
Number of Residues19
Detailsbinding site for residue XG4 E 705
ChainResidue
EGLN149
ELEU150
EARG164
EHIS167
EASP207
EHIS210
EHIS215
EHIS233
EASP311
ELYS312
ETYR315
EASP319
EARG366
EHIS370
ETYR374
EGLN375
EFE701
EMG702
EMG703

site_idAG2
Number of Residues14
Detailsbinding site for residue CZF E 706
ChainResidue
ELYS116
EVAL117
EILE118
EASN137
EGLN142
EARG145
EPHE165
EMG704
FTYR155
FVAL156
FVAL378
FARG451
GLYS523
GXG4701

site_idAG3
Number of Residues4
Detailsbinding site for residue SO4 E 707
ChainResidue
EARG305
EARG348
EHIS517
EARG531

site_idAG4
Number of Residues15
Detailsbinding site for residue XG4 E 708
ChainResidue
EARG333
EARG352
ELYS354
EASN358
ELYS523
GVAL117
GASN119
GMG705
GCZF707
HVAL156
HPHE157
HILE325
HARG372
HHIS376
HLYS377

site_idAG5
Number of Residues7
Detailsbinding site for residue FE F 701
ChainResidue
FARG164
FHIS167
FHIS206
FASP207
FASP311
FMG702
FXG4705

site_idAG6
Number of Residues6
Detailsbinding site for residue MG F 702
ChainResidue
FHIS206
FASP207
FHIS233
FASP311
FFE701
FXG4705

site_idAG7
Number of Residues3
Detailsbinding site for residue MG F 703
ChainResidue
FASP309
FLYS312
FXG4705

site_idAG8
Number of Residues2
Detailsbinding site for residue MG F 704
ChainResidue
FCZF706
HXG4701

site_idAG9
Number of Residues18
Detailsbinding site for residue XG4 F 705
ChainResidue
FGLN149
FLEU150
FARG164
FHIS167
FASP207
FHIS210
FHIS215
FHIS233
FASP311
FLYS312
FTYR315
FASP319
FARG366
FTYR374
FGLN375
FFE701
FMG702
FMG703

site_idAH1
Number of Residues15
Detailsbinding site for residue CZF F 706
ChainResidue
ETYR155
EVAL156
EVAL378
EARG451
ELYS455
FLYS116
FVAL117
FILE118
FASN137
FGLN142
FARG145
FPHE165
FMG704
HLYS523
HXG4701

site_idAH2
Number of Residues4
Detailsbinding site for residue SO4 F 707
ChainResidue
FARG305
FARG348
FHIS517
FARG531

site_idAH3
Number of Residues16
Detailsbinding site for residue XG4 F 708
ChainResidue
FASP330
FARG333
FARG352
FLYS354
FASN358
FLYS523
GVAL156
GPHE157
GARG372
GHIS376
GLYS377
HVAL117
HASN119
HHIS125
HMG705
HCZF707

site_idAH4
Number of Residues17
Detailsbinding site for residue XG4 G 701
ChainResidue
EVAL117
EASN119
EHIS125
EMG704
ECZF706
FVAL156
FPHE157
FGLY324
FARG372
FHIS376
FLYS377
GASP330
GARG333
GARG352
GLYS354
GASN358
GLYS523

site_idAH5
Number of Residues7
Detailsbinding site for residue FE G 702
ChainResidue
GARG164
GHIS167
GHIS206
GASP207
GASP311
GMG703
GXG4706

site_idAH6
Number of Residues6
Detailsbinding site for residue MG G 703
ChainResidue
GHIS206
GASP207
GHIS233
GASP311
GFE702
GXG4706

site_idAH7
Number of Residues3
Detailsbinding site for residue MG G 704
ChainResidue
GASP309
GLYS312
GXG4706

site_idAH8
Number of Residues2
Detailsbinding site for residue MG G 705
ChainResidue
EXG4708
GCZF707

site_idAH9
Number of Residues18
Detailsbinding site for residue XG4 G 706
ChainResidue
GGLN149
GLEU150
GARG164
GHIS167
GASP207
GHIS210
GHIS215
GHIS233
GASP311
GLYS312
GTYR315
GASP319
GARG366
GTYR374
GGLN375
GFE702
GMG703
GMG704

site_idAI1
Number of Residues15
Detailsbinding site for residue CZF G 707
ChainResidue
ELYS523
EXG4708
GLYS116
GVAL117
GILE118
GASN137
GGLN142
GARG145
GPHE165
GMG705
HTYR155
HVAL156
HVAL378
HARG451
HLYS455

site_idAI2
Number of Residues4
Detailsbinding site for residue SO4 G 708
ChainResidue
GARG305
GARG348
GHIS517
GARG531

site_idAI3
Number of Residues17
Detailsbinding site for residue XG4 H 701
ChainResidue
EVAL156
EPHE157
EGLY324
EARG372
EHIS376
ELYS377
FVAL117
FASN119
FHIS125
FMG704
FCZF706
HASP330
HARG333
HARG352
HLYS354
HASN358
HLYS523

site_idAI4
Number of Residues7
Detailsbinding site for residue FE H 702
ChainResidue
HARG164
HHIS167
HHIS206
HASP207
HASP311
HMG703
HXG4706

site_idAI5
Number of Residues5
Detailsbinding site for residue MG H 703
ChainResidue
HHIS206
HASP207
HHIS233
HFE702
HXG4706

site_idAI6
Number of Residues3
Detailsbinding site for residue MG H 704
ChainResidue
HASP309
HLYS312
HXG4706

site_idAI7
Number of Residues2
Detailsbinding site for residue MG H 705
ChainResidue
FXG4708
HCZF707

site_idAI8
Number of Residues18
Detailsbinding site for residue XG4 H 706
ChainResidue
HGLN149
HLEU150
HARG164
HHIS167
HASP207
HHIS210
HHIS215
HHIS233
HASP311
HLYS312
HTYR315
HASP319
HARG366
HTYR374
HGLN375
HFE702
HMG703
HMG704

site_idAI9
Number of Residues15
Detailsbinding site for residue CZF H 707
ChainResidue
FLYS523
FXG4708
GTYR155
GVAL156
GLYS377
GVAL378
GARG451
HLYS116
HVAL117
HILE118
HASN137
HGLN142
HARG145
HPHE165
HMG705

site_idAJ1
Number of Residues4
Detailsbinding site for residue SO4 H 708
ChainResidue
HARG305
HARG348
HHIS517
HARG531

site_idAJ2
Number of Residues7
Detailsbinding site for residue FE I 701
ChainResidue
IARG164
IHIS167
IHIS206
IASP207
IASP311
IMG702
IXG4705

site_idAJ3
Number of Residues5
Detailsbinding site for residue MG I 702
ChainResidue
IHIS206
IASP207
IHIS233
IFE701
IXG4705

site_idAJ4
Number of Residues2
Detailsbinding site for residue MG I 703
ChainResidue
IASP309
IXG4705

site_idAJ5
Number of Residues2
Detailsbinding site for residue MG I 704
ChainResidue
JCZF701
KXG4701

site_idAJ6
Number of Residues19
Detailsbinding site for residue XG4 I 705
ChainResidue
IGLN149
ILEU150
IARG164
IHIS167
IASP207
IHIS210
IHIS215
IHIS233
IASP311
ILYS312
ITYR315
IASP319
IARG366
IHIS370
ITYR374
IGLN375
IFE701
IMG702
IMG703

site_idAJ7
Number of Residues4
Detailsbinding site for residue SO4 I 706
ChainResidue
IARG305
IARG348
IHIS517
IARG531

site_idAJ8
Number of Residues16
Detailsbinding site for residue XG4 I 707
ChainResidue
IVAL156
IPHE157
IGLY324
IILE325
IARG372
IHIS376
ILYS377
JVAL117
JASN119
JMG705
JCZF707
LARG333
LARG352
LLYS354
LASN358
LLYS523

site_idAJ9
Number of Residues17
Detailsbinding site for residue XG4 I 708
ChainResidue
IASP330
IARG333
IARG352
ILYS354
IASN358
ILYS523
KVAL117
KASN119
KHIS125
KMG705
KCZF707
LVAL156
LPHE157
LGLY324
LARG372
LHIS376
LLYS377

site_idAK1
Number of Residues14
Detailsbinding site for residue CZF J 701
ChainResidue
ILYS116
IVAL117
IILE118
IASN137
IGLN142
IARG145
IPHE165
IMG704
JTYR155
JVAL156
JVAL378
JARG451
KLYS523
KXG4701

site_idAK2
Number of Residues7
Detailsbinding site for residue FE J 702
ChainResidue
JARG164
JHIS167
JHIS206
JASP207
JASP311
JMG703
JXG4706

site_idAK3
Number of Residues4
Detailsbinding site for residue MG J 703
ChainResidue
JASP207
JHIS233
JFE702
JXG4706

site_idAK4
Number of Residues3
Detailsbinding site for residue MG J 704
ChainResidue
JASP309
JLYS312
JXG4706

site_idAK5
Number of Residues2
Detailsbinding site for residue MG J 705
ChainResidue
IXG4707
JCZF707

site_idAK6
Number of Residues18
Detailsbinding site for residue XG4 J 706
ChainResidue
JGLN149
JLEU150
JARG164
JHIS167
JASP207
JHIS215
JHIS233
JASP311
JLYS312
JTYR315
JASP319
JARG366
JHIS370
JTYR374
JGLN375
JFE702
JMG703
JMG704

site_idAK7
Number of Residues14
Detailsbinding site for residue CZF J 707
ChainResidue
ITYR155
IVAL156
IVAL378
IARG451
IXG4707
JLYS116
JVAL117
JILE118
JASN137
JGLN142
JARG145
JPHE165
JMG705
LLYS523

site_idAK8
Number of Residues4
Detailsbinding site for residue SO4 J 708
ChainResidue
JARG305
JARG348
JHIS517
JARG531

site_idAK9
Number of Residues19
Detailsbinding site for residue XG4 J 709
ChainResidue
JASP330
JARG333
JARG352
JLYS354
JASN358
JLYS523
KVAL156
KPHE157
KGLY324
KILE325
KARG372
KHIS376
KLYS377
LVAL117
LILE118
LASN119
LHIS125
LMG704
LCZF706

site_idAL1
Number of Residues17
Detailsbinding site for residue XG4 K 701
ChainResidue
IVAL117
IASN119
IHIS125
IMG704
JVAL156
JPHE157
JGLY324
JARG372
JHIS376
JLYS377
JCZF701
KASP330
KARG333
KARG352
KLYS354
KASN358
KLYS523

site_idAL2
Number of Residues7
Detailsbinding site for residue FE K 702
ChainResidue
KARG164
KHIS167
KHIS206
KASP207
KASP311
KMG703
KXG4706

site_idAL3
Number of Residues5
Detailsbinding site for residue MG K 703
ChainResidue
KHIS206
KASP207
KHIS233
KFE702
KXG4706

site_idAL4
Number of Residues3
Detailsbinding site for residue MG K 704
ChainResidue
KASP309
KLYS312
KXG4706

site_idAL5
Number of Residues2
Detailsbinding site for residue MG K 705
ChainResidue
IXG4708
KCZF707

site_idAL6
Number of Residues19
Detailsbinding site for residue XG4 K 706
ChainResidue
KGLN149
KLEU150
KARG164
KHIS167
KASP207
KHIS210
KHIS215
KHIS233
KASP311
KLYS312
KTYR315
KASP319
KARG366
KHIS370
KTYR374
KGLN375
KFE702
KMG703
KMG704

site_idAL7
Number of Residues14
Detailsbinding site for residue CZF K 707
ChainResidue
ILYS523
IXG4708
KLYS116
KVAL117
KILE118
KASN137
KGLN142
KARG145
KPHE165
KMG705
LTYR155
LVAL156
LVAL378
LARG451

site_idAL8
Number of Residues4
Detailsbinding site for residue SO4 K 708
ChainResidue
KARG305
KARG348
KHIS517
KARG531

site_idAL9
Number of Residues7
Detailsbinding site for residue FE L 701
ChainResidue
LARG164
LHIS167
LHIS206
LASP207
LASP311
LMG702
LXG4705

site_idAM1
Number of Residues6
Detailsbinding site for residue MG L 702
ChainResidue
LHIS206
LASP207
LHIS233
LASP311
LFE701
LXG4705

site_idAM2
Number of Residues3
Detailsbinding site for residue MG L 703
ChainResidue
LASP309
LLYS312
LXG4705

site_idAM3
Number of Residues2
Detailsbinding site for residue MG L 704
ChainResidue
JXG4709
LCZF706

site_idAM4
Number of Residues19
Detailsbinding site for residue XG4 L 705
ChainResidue
LGLN149
LLEU150
LARG164
LHIS167
LASP207
LHIS210
LHIS215
LHIS233
LASP311
LLYS312
LTYR315
LASP319
LARG366
LHIS370
LTYR374
LGLN375
LFE701
LMG702
LMG703

site_idAM5
Number of Residues15
Detailsbinding site for residue CZF L 706
ChainResidue
JLYS523
JXG4709
KTYR155
KVAL156
KVAL378
KARG451
KLYS455
LLYS116
LVAL117
LILE118
LASN137
LGLN142
LARG145
LPHE165
LMG704

site_idAM6
Number of Residues4
Detailsbinding site for residue SO4 L 707
ChainResidue
LARG305
LARG348
LHIS517
LARG531

site_idAM7
Number of Residues6
Detailsbinding site for residue FE M 701
ChainResidue
MARG164
MHIS167
MHIS206
MASP207
MASP311
MXG4705

site_idAM8
Number of Residues4
Detailsbinding site for residue MG M 702
ChainResidue
MHIS206
MASP207
MHIS233
MXG4705

site_idAM9
Number of Residues2
Detailsbinding site for residue MG M 703
ChainResidue
MASP309
MXG4705

site_idAN1
Number of Residues3
Detailsbinding site for residue MG M 704
ChainResidue
MLYS116
MCZF706
OXG4701

site_idAN2
Number of Residues18
Detailsbinding site for residue XG4 M 705
ChainResidue
MGLN149
MLEU150
MARG164
MHIS167
MASP207
MHIS210
MHIS215
MHIS233
MASP311
MLYS312
MTYR315
MASP319
MARG366
MTYR374
MGLN375
MFE701
MMG702
MMG703

site_idAN3
Number of Residues15
Detailsbinding site for residue CZF M 706
ChainResidue
MLYS116
MVAL117
MILE118
MASN137
MGLN142
MARG145
MPHE165
MMG704
NTYR155
NVAL156
NVAL378
NARG451
NLYS455
OLYS523
OXG4701

site_idAN4
Number of Residues4
Detailsbinding site for residue SO4 M 707
ChainResidue
MARG305
MARG348
MHIS517
MARG531

site_idAN5
Number of Residues16
Detailsbinding site for residue XG4 M 708
ChainResidue
MARG333
MARG352
MLYS354
MASN358
MLYS523
OVAL117
OASN119
OHIS125
OMG705
OCZF707
PVAL156
PPHE157
PGLY324
PARG372
PHIS376
PLYS377

site_idAN6
Number of Residues7
Detailsbinding site for residue FE N 701
ChainResidue
NARG164
NHIS167
NHIS206
NASP207
NASP311
NMG702
NXG4705

site_idAN7
Number of Residues5
Detailsbinding site for residue MG N 702
ChainResidue
NHIS206
NASP207
NHIS233
NFE701
NXG4705

site_idAN8
Number of Residues3
Detailsbinding site for residue MG N 703
ChainResidue
NASP309
NLYS312
NXG4705

site_idAN9
Number of Residues2
Detailsbinding site for residue MG N 704
ChainResidue
NCZF706
PXG4701

site_idAO1
Number of Residues19
Detailsbinding site for residue XG4 N 705
ChainResidue
NGLN149
NLEU150
NARG164
NHIS167
NASP207
NHIS210
NHIS215
NHIS233
NASP311
NLYS312
NTYR315
NASP319
NARG366
NHIS370
NTYR374
NGLN375
NFE701
NMG702
NMG703

site_idAO2
Number of Residues14
Detailsbinding site for residue CZF N 706
ChainResidue
MTYR155
MVAL156
MVAL378
MARG451
NLYS116
NVAL117
NILE118
NASN137
NGLN142
NARG145
NPHE165
NMG704
PLYS523
PXG4701

site_idAO3
Number of Residues3
Detailsbinding site for residue SO4 N 707
ChainResidue
NARG305
NARG348
NHIS517

site_idAO4
Number of Residues17
Detailsbinding site for residue XG4 N 708
ChainResidue
NASP330
NARG333
NARG352
NLYS354
NASN358
NLYS523
OVAL156
OPHE157
OGLY324
OARG372
OHIS376
OLYS377
PILE118
PASN119
PHIS125
PMG705
PCZF707

site_idAO5
Number of Residues18
Detailsbinding site for residue XG4 O 701
ChainResidue
MVAL117
MASN119
MHIS125
MMG704
MCZF706
NVAL156
NPHE157
NGLY324
NARG372
NHIS376
NLYS377
NVAL378
OASP330
OARG333
OARG352
OLYS354
OASN358
OLYS523

site_idAO6
Number of Residues7
Detailsbinding site for residue FE O 702
ChainResidue
OARG164
OHIS167
OHIS206
OASP207
OASP311
OMG703
OXG4706

site_idAO7
Number of Residues5
Detailsbinding site for residue MG O 703
ChainResidue
OHIS206
OASP207
OHIS233
OFE702
OXG4706

site_idAO8
Number of Residues2
Detailsbinding site for residue MG O 704
ChainResidue
OASP309
OXG4706

site_idAO9
Number of Residues2
Detailsbinding site for residue MG O 705
ChainResidue
MXG4708
OCZF707

site_idAP1
Number of Residues19
Detailsbinding site for residue XG4 O 706
ChainResidue
OGLN149
OLEU150
OARG164
OHIS167
OASP207
OHIS210
OHIS215
OHIS233
OASP311
OLYS312
OTYR315
OASP319
OARG366
OHIS370
OTYR374
OGLN375
OFE702
OMG703
OMG704

site_idAP2
Number of Residues14
Detailsbinding site for residue CZF O 707
ChainResidue
MLYS523
MXG4708
OLYS116
OVAL117
OILE118
OASN137
OGLN142
OARG145
OPHE165
OMG705
PTYR155
PVAL156
PVAL378
PARG451

site_idAP3
Number of Residues4
Detailsbinding site for residue SO4 O 708
ChainResidue
OARG305
OARG348
OHIS517
OARG531

site_idAP4
Number of Residues16
Detailsbinding site for residue XG4 P 701
ChainResidue
MVAL156
MPHE157
MARG372
MHIS376
MLYS377
NVAL117
NASN119
NHIS125
NMG704
NCZF706
PASP330
PARG333
PARG352
PLYS354
PASN358
PLYS523

site_idAP5
Number of Residues7
Detailsbinding site for residue FE P 702
ChainResidue
PARG164
PHIS167
PHIS206
PASP207
PASP311
PMG703
PXG4706

site_idAP6
Number of Residues6
Detailsbinding site for residue MG P 703
ChainResidue
PHIS206
PASP207
PHIS233
PASP311
PFE702
PXG4706

site_idAP7
Number of Residues2
Detailsbinding site for residue MG P 704
ChainResidue
PASP309
PXG4706

site_idAP8
Number of Residues2
Detailsbinding site for residue MG P 705
ChainResidue
NXG4708
PCZF707

site_idAP9
Number of Residues19
Detailsbinding site for residue XG4 P 706
ChainResidue
PGLN149
PLEU150
PARG164
PHIS167
PASP207
PHIS210
PHIS215
PHIS233
PASP311
PLYS312
PTYR315
PASP319
PARG366
PHIS370
PTYR374
PGLN375
PFE702
PMG703
PMG704

site_idAQ1
Number of Residues15
Detailsbinding site for residue CZF P 707
ChainResidue
NLYS523
NXG4708
OTYR155
OVAL156
OVAL378
OARG451
OLYS455
PLYS116
PVAL117
PILE118
PASN137
PGLN142
PARG145
PPHE165
PMG705

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues16
DetailsACT_SITE: ACT_SITE => ECO:0000305|PubMed:22056990
ChainResidueDetails
AHIS233
BHIS233
CHIS233
DHIS233
EHIS233
FHIS233
GHIS233
HHIS233
IHIS233
JHIS233
KHIS233
LHIS233
MHIS233
NHIS233
OHIS233
PHIS233

site_idSWS_FT_FI2
Number of Residues96
DetailsBINDING: in other chain => ECO:0000269|PubMed:24141705, ECO:0000269|PubMed:24217394, ECO:0000269|PubMed:25267621, ECO:0000269|PubMed:25288794, ECO:0000269|PubMed:25760601, ECO:0000269|PubMed:26294762, ECO:0000269|PubMed:26431200
ChainResidueDetails
CASN358
CLYS523
DLYS116
DASN137
DARG333
DARG352
DASN358
DLYS523
ELYS116
EASN137
EARG333
EARG352
EASN358
ELYS523
FLYS116
FASN137
FARG333
FARG352
FASN358
FLYS523
GLYS116
GASN137
GARG333
GARG352
GASN358
GLYS523
HLYS116
HASN137
HARG333
HARG352
HASN358
HLYS523
ILYS116
IASN137
IARG333
IARG352
IASN358
ILYS523
JLYS116
JASN137
JARG333
JARG352
JASN358
JLYS523
KLYS116
KASN137
KARG333
KARG352
KASN358
KLYS523
LLYS116
LASN137
LARG333
LARG352
LASN358
LLYS523
MLYS116
MASN137
MARG333
MARG352
MASN358
MLYS523
NLYS116
NASN137
NARG333
NARG352
NASN358
NLYS523
OLYS116
OASN137
OARG333
OARG352
OASN358
OLYS523
PLYS116
PASN137
PARG333
PARG352
PASN358
PLYS523
ALYS116
AASN137
AARG333
AARG352
AASN358
ALYS523
BLYS116
BASN137
BARG333
BARG352
BASN358
BLYS523
CLYS116
CASN137
CARG333
CARG352

site_idSWS_FT_FI3
Number of Residues80
DetailsBINDING: BINDING => ECO:0000269|PubMed:24141705, ECO:0000269|PubMed:24217394, ECO:0000269|PubMed:25267621, ECO:0000269|PubMed:25288794, ECO:0000269|PubMed:25760601, ECO:0000269|PubMed:26294762, ECO:0000269|PubMed:26431200
ChainResidueDetails
DHIS376
DLYS377
DARG451
DLYS455
EASN119
EHIS376
ELYS377
EARG451
ELYS455
FASN119
FHIS376
FLYS377
FARG451
FLYS455
GASN119
GHIS376
GLYS377
GARG451
GLYS455
HASN119
HHIS376
HLYS377
HARG451
HLYS455
IASN119
IHIS376
ILYS377
IARG451
ILYS455
JASN119
JHIS376
JLYS377
JARG451
JLYS455
KASN119
KHIS376
KLYS377
KARG451
KLYS455
LASN119
LHIS376
LLYS377
LARG451
LLYS455
MASN119
MHIS376
MLYS377
MARG451
MLYS455
NASN119
NHIS376
NLYS377
NARG451
NLYS455
OASN119
OHIS376
OLYS377
OARG451
OLYS455
PASN119
PHIS376
PLYS377
PARG451
PLYS455
AHIS376
ALYS377
AARG451
ALYS455
BASN119
BHIS376
BLYS377
BARG451
BLYS455
CASN119
CHIS376
CLYS377
CARG451
CLYS455
DASN119
AASN119

site_idSWS_FT_FI4
Number of Residues128
DetailsBINDING: BINDING => ECO:0000269|PubMed:24141705
ChainResidueDetails
EGLN149
EARG164
EHIS210
EASP309
ETYR315
EASP319
EARG366
EHIS370
FGLN149
FARG164
FHIS210
FASP309
FTYR315
FASP319
FARG366
FHIS370
GGLN149
GARG164
GHIS210
GASP309
GTYR315
GASP319
GARG366
GHIS370
HGLN149
HARG164
HHIS210
HASP309
HTYR315
HASP319
HARG366
HHIS370
IGLN149
IARG164
IHIS210
IASP309
ITYR315
IASP319
IARG366
IHIS370
JGLN149
JARG164
JHIS210
JASP309
JTYR315
JASP319
JARG366
JHIS370
KGLN149
KARG164
KHIS210
KASP309
KTYR315
KASP319
KARG366
KHIS370
LGLN149
LARG164
LHIS210
LASP309
LTYR315
LASP319
LARG366
LHIS370
MGLN149
MARG164
MHIS210
MASP309
MTYR315
MASP319
MARG366
MHIS370
NGLN149
NARG164
NHIS210
NASP309
NTYR315
NASP319
NARG366
NHIS370
OGLN149
OARG164
OHIS210
OASP309
OTYR315
OASP319
OARG366
OHIS370
PGLN149
PARG164
PHIS210
PASP309
PTYR315
PASP319
PARG366
PHIS370
AHIS210
AASP309
ATYR315
AASP319
AARG366
AHIS370
BGLN149
BARG164
BHIS210
BASP309
BTYR315
BASP319
BARG366
BHIS370
CGLN149
CARG164
CHIS210
CASP309
CTYR315
CASP319
CARG366
CHIS370
DGLN149
DARG164
DHIS210
DASP309
DTYR315
DASP319
DARG366
DHIS370
AGLN149
AARG164

site_idSWS_FT_FI5
Number of Residues64
DetailsBINDING: BINDING => ECO:0000269|PubMed:24141705, ECO:0000269|PubMed:24217394, ECO:0000269|PubMed:25288794, ECO:0000269|PubMed:25760601, ECO:0000269|PubMed:26431200
ChainResidueDetails
IHIS167
IHIS206
IASP207
IASP311
JHIS167
JHIS206
JASP207
JASP311
KHIS167
KHIS206
KASP207
KASP311
LHIS167
LHIS206
LASP207
LASP311
MHIS167
MHIS206
MASP207
MASP311
NHIS167
NHIS206
NASP207
NASP311
OHIS167
OHIS206
OASP207
OASP311
PHIS167
PHIS206
PASP207
PASP311
AASP207
AASP311
BHIS167
BHIS206
BASP207
BASP311
CHIS167
CHIS206
CASP207
CASP311
DHIS167
DHIS206
DASP207
DASP311
EHIS167
EHIS206
EASP207
EASP311
FHIS167
FHIS206
FASP207
FASP311
GHIS167
GHIS206
GASP207
GASP311
HHIS167
HHIS206
HASP207
HASP311
AHIS167
AHIS206

site_idSWS_FT_FI6
Number of Residues16
DetailsMOD_RES: Phosphothreonine; by CDK1 => ECO:0000269|PubMed:23601106, ECO:0000269|PubMed:23602554, ECO:0000269|PubMed:26294762, ECO:0000269|PubMed:26431200, ECO:0000269|PubMed:29610582, ECO:0000269|PubMed:29670289, ECO:0007744|PubMed:17081983, ECO:0007744|PubMed:18669648, ECO:0007744|PubMed:18691976, ECO:0007744|PubMed:19369195, ECO:0007744|PubMed:20068231, ECO:0007744|PubMed:23186163, ECO:0007744|PubMed:24275569
ChainResidueDetails
BTHR592
CTHR592
DTHR592
ETHR592
FTHR592
GTHR592
HTHR592
ITHR592
JTHR592
KTHR592
LTHR592
MTHR592
NTHR592
OTHR592
PTHR592
ATHR592

site_idSWS_FT_FI7
Number of Residues80
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
DLYS469
DLYS492
DLYS622
ELYS467
ELYS469
ELYS492
ELYS622
FLYS467
FLYS469
FLYS492
FLYS622
GLYS467
GLYS469
GLYS492
GLYS622
HLYS467
HLYS469
HLYS492
HLYS622
ILYS467
ILYS469
ILYS492
ILYS622
JLYS467
JLYS469
JLYS492
JLYS622
KLYS467
KLYS469
KLYS492
KLYS622
LLYS467
LLYS469
LLYS492
LLYS622
MLYS467
MLYS469
MLYS492
MLYS622
NLYS467
NLYS469
NLYS492
NLYS622
OLYS467
OLYS469
OLYS492
OLYS622
PLYS467
PLYS469
PLYS492
PLYS622
ALYS469
ALYS492
ALYS622
BLYS467
BLYS469
BLYS492
BLYS622
CLYS467
CLYS469
CLYS492
CLYS622
DLYS467
ALYS467

221051

PDB entries from 2024-06-12

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