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6SCM

SOS1 in Complex with Inhibitor BI-3406

Functional Information from GO Data
ChainGOidnamespacecontents
A0005085molecular_functionguanyl-nucleotide exchange factor activity
A0007264biological_processsmall GTPase-mediated signal transduction
Functional Information from PDB Data
site_idAC1
Number of Residues5
Detailsbinding site for residue IMD A 1101
ChainResidue
ATYR884
AASP887
APHE890
AIMD1102
AL7H1108

site_idAC2
Number of Residues4
Detailsbinding site for residue IMD A 1102
ChainResidue
ATYR884
AGLU902
AIMD1101
AL7H1108

site_idAC3
Number of Residues4
Detailsbinding site for residue EDO A 1103
ChainResidue
APHE648
AGLU649
ATHR720
AHOH1301

site_idAC4
Number of Residues7
Detailsbinding site for residue EDO A 1104
ChainResidue
AGLY943
AASN944
ATYR1008
AASN1011
ALYS1012
AGLU1015
AHOH1273

site_idAC5
Number of Residues7
Detailsbinding site for residue EDO A 1105
ChainResidue
ASER633
AVAL805
AGLY806
AGLU941
AGLU946
AARG961
ALYS1022

site_idAC6
Number of Residues6
Detailsbinding site for residue EDO A 1106
ChainResidue
AARG625
AGLU664
AASN691
AARG694
AHIS695
AHOH1320

site_idAC7
Number of Residues3
Detailsbinding site for residue EDO A 1107
ChainResidue
ASER876
AASN879
ATYR912

site_idAC8
Number of Residues11
Detailsbinding site for residue L7H A 1108
ChainResidue
AGLU590
AASN591
AMET878
AASN879
ATYR884
APHE890
ALYS898
AGLU902
AHIS905
AIMD1101
AIMD1102

Functional Information from PROSITE/UniProt
site_idPS00720
Number of Residues34
DetailsRASGEF Ras Guanine-nucleotide exchange factors domain signature. VPFfGiyLtNIlkteegnpevlkrhgkel.................INFsK
ChainResidueDetails
AVAL927-LYS960

221051

PDB entries from 2024-06-12

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