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6SAJ

Crystal Structure of BRD4(1) bound to inhibitor BUX6 (12)

Functional Information from PDB Data
site_idAC1
Number of Residues5
Detailsbinding site for residue BU3 A 201
ChainResidue
AMET149
AL2Z204
AHOH302
AHOH323
AHOH384

site_idAC2
Number of Residues6
Detailsbinding site for residue BU3 A 202
ChainResidue
AASN135
AHOH386
AILE100
AILE101
ALYS102
ATHR103

site_idAC3
Number of Residues5
Detailsbinding site for residue BU3 A 203
ChainResidue
ALYS112
AGLU115
AASN116
AASP145
AHOH310

site_idAC4
Number of Residues15
Detailsbinding site for residue L2Z A 204
ChainResidue
ALYS57
AGLN59
ATRP81
APRO82
AVAL87
ALYS91
ALEU92
ALYS102
AASN117
ATYR139
AASN140
AILE146
ABU3201
AHOH325
AHOH351

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues106
DetailsDomain: {"description":"Bromo 1","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues1
DetailsSite: {"description":"Acetylated histone binding","evidences":[{"source":"PubMed","id":"22464331","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues2
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2)","evidences":[{"source":"PubMed","id":"28112733","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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