6S60
Crystal structure of hTEAD2 in complex with a trisubstituted pyrazole inhibitor
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 7 |
Details | binding site for residue MYR A 501 |
Chain | Residue |
A | ALA235 |
A | ALA304 |
A | LYS357 |
A | MET379 |
A | CYS380 |
A | LEU403 |
A | ILE408 |
site_id | AC2 |
Number of Residues | 5 |
Details | binding site for residue KX8 B 502 |
Chain | Residue |
B | LYS352 |
B | VAL354 |
B | TYR382 |
A | TYR397 |
B | SER349 |
site_id | AC3 |
Number of Residues | 10 |
Details | binding site for Di-peptide MYR B 501 and CYS B 380 |
Chain | Residue |
B | ALA235 |
B | SER345 |
B | PRO378 |
B | MET379 |
B | GLU381 |
B | TYR382 |
B | LEU383 |
B | VAL384 |
B | ILE408 |
B | PHE428 |