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6S60

Crystal structure of hTEAD2 in complex with a trisubstituted pyrazole inhibitor

Functional Information from PDB Data
site_idAC1
Number of Residues7
Detailsbinding site for residue MYR A 501
ChainResidue
AALA235
AALA304
ALYS357
AMET379
ACYS380
ALEU403
AILE408

site_idAC2
Number of Residues5
Detailsbinding site for residue KX8 B 502
ChainResidue
BLYS352
BVAL354
BTYR382
ATYR397
BSER349

site_idAC3
Number of Residues10
Detailsbinding site for Di-peptide MYR B 501 and CYS B 380
ChainResidue
BALA235
BSER345
BPRO378
BMET379
BGLU381
BTYR382
BLEU383
BVAL384
BILE408
BPHE428

221051

PDB entries from 2024-06-12

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