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6QDE

Leishmania major N-myristoyltransferase in complex with thienopyrimidine inhibitor IMP-0000877

Functional Information from GO Data
ChainGOidnamespacecontents
A0004379molecular_functionglycylpeptide N-tetradecanoyltransferase activity
A0005829cellular_componentcytosol
A0006499biological_processN-terminal protein myristoylation
A0016740molecular_functiontransferase activity
A0016746molecular_functionacyltransferase activity
A0046872molecular_functionmetal ion binding
A0072657biological_processprotein localization to membrane
Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue MG A 501
ChainResidue
ALEU175
AGLU177
ALYS178
AARG179
ALEU180
AMYA504

site_idAC2
Number of Residues11
Detailsbinding site for residue HWW A 502
ChainResidue
AGLY205
ATYR217
AILE328
ATYR345
AHIS398
AMET420
ALEU421
AHWW503
APHE90
AASN167
ATHR203

site_idAC3
Number of Residues16
Detailsbinding site for residue HWW A 503
ChainResidue
AVAL81
AGLU82
AASP83
AASP84
AMET87
APHE88
APHE90
APHE232
ASER330
ATYR345
AASN376
AASP396
AHWW502
AHOH611
AHOH766
AHOH887

site_idAC4
Number of Residues35
Detailsbinding site for residue MYA A 504
ChainResidue
AHIS12
AALA13
APHE14
ATRP15
ATYR80
AVAL81
APHE168
ALEU169
ACYS170
AVAL171
AARG176
AGLU177
ALYS178
AARG179
ALEU180
AALA181
APRO182
ATHR189
AVAL192
ATRP198
ATYR202
ATHR203
ALEU208
ATYR404
AMG501
AHOH650
AHOH661
AHOH665
AHOH668
AHOH703
AHOH825
AHOH839
AHOH871
AHOH878
AHOH975

Functional Information from PROSITE/UniProt
site_idPS00975
Number of Residues9
DetailsNMT_1 Myristoyl-CoA:protein N-myristoyltransferase signature 1. EINFLCvHK
ChainResidueDetails
AGLU165-LYS173

site_idPS00976
Number of Residues7
DetailsNMT_2 Myristoyl-CoA:protein N-myristoyltransferase signature 2. KFGaGDG
ChainResidueDetails
ALYS391-GLY397

247947

PDB entries from 2026-01-21

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