6Q6O
RORCVAR2 (RORGT, 264-499) IN COMPLEX WITH COMPOUND 2 AT 2.3A: Identification of N-aryl imidazoles as potent and selective RORgt inhibitors
Functional Information from GO Data
Functional Information from PDB Data
| site_id | AC1 |
| Number of Residues | 10 |
| Details | binding site for residue HKE A 501 |
| Chain | Residue |
| A | CYS320 |
| A | LEU483 |
| A | HIS323 |
| A | LEU324 |
| A | VAL361 |
| A | PHE378 |
| A | PHE388 |
| A | ILE397 |
| A | ILE400 |
| A | HIS479 |
| site_id | AC2 |
| Number of Residues | 5 |
| Details | binding site for residue CHD A 502 |
| Chain | Residue |
| A | GLN329 |
| A | GLU333 |
| A | LYS336 |
| A | LYS354 |
| A | CHD503 |
| site_id | AC3 |
| Number of Residues | 5 |
| Details | binding site for residue CHD A 503 |
| Chain | Residue |
| A | THR325 |
| A | LEU483 |
| A | GLN484 |
| A | GLN487 |
| A | CHD502 |






