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6Q6M

RORCVAR2 (RORGT, 264-499) IN COMPLEX WITH COMPOUND 1: Identification of N-aryl imidazoles as potent and selective RORgt inhibitors

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue HJW A 501
ChainResidue
ACYS320
AHIS479
AHIS323
ALEU324
AVAL361
ALEU362
APHE378
APHE388
ALEU391
AILE397

224201

PDB entries from 2024-08-28

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