6P9F
Crystal structure of RAR-related orphan receptor C (NHIS-RORGT(244-487)-L6-SRC1(678-692)) in complex with a phenyl (3-phenylpyrrolidin-3-yl)sulfone inhibitor
Functional Information from GO Data
Chain | GOid | namespace | contents |
A | 0003677 | molecular_function | DNA binding |
A | 0004879 | molecular_function | nuclear receptor activity |
A | 0005634 | cellular_component | nucleus |
A | 0006355 | biological_process | regulation of DNA-templated transcription |
B | 0003677 | molecular_function | DNA binding |
B | 0004879 | molecular_function | nuclear receptor activity |
B | 0005634 | cellular_component | nucleus |
B | 0006355 | biological_process | regulation of DNA-templated transcription |
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 20 |
Details | binding site for residue O5A A 4000 |
Chain | Residue |
A | GLN286 |
A | VAL376 |
A | PHE378 |
A | PHE388 |
A | LEU391 |
A | LEU396 |
A | ILE397 |
A | ILE400 |
A | PHE401 |
A | HIS479 |
A | HOH4101 |
A | LEU287 |
A | HOH4105 |
A | CYS320 |
A | HIS323 |
A | LEU324 |
A | ALA327 |
A | ARG364 |
A | MET365 |
A | ARG367 |
site_id | AC2 |
Number of Residues | 18 |
Details | binding site for residue O5A B 4000 |
Chain | Residue |
B | GLN286 |
B | LEU287 |
B | CYS320 |
B | HIS323 |
B | LEU324 |
B | MET358 |
B | ARG364 |
B | MET365 |
B | ARG367 |
B | VAL376 |
B | PHE378 |
B | PHE388 |
B | LEU396 |
B | ILE397 |
B | ILE400 |
B | PHE401 |
B | HIS479 |
B | HOH4103 |