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6P54

Crystal structure of transpeptidase domain of PBP2 from Neisseria gonorrhoeae acylated by ceftriaxone

Functional Information from GO Data
ChainGOidnamespacecontents
A0008658molecular_functionpenicillin binding
B0008658molecular_functionpenicillin binding
Functional Information from PDB Data
site_idAC1
Number of Residues17
Detailsbinding site for residue NZV A 600
ChainResidue
AGLU307
ATHR500
AALA501
AARG502
ATYR509
AHIS514
ATYR543
ATYR544
AHOH734
ASER310
ATHR347
ASER362
AASN364
APHE420
ATYR422
ATHR498
AGLY499

site_idAC2
Number of Residues6
Detailsbinding site for residue 9F2 B 602
ChainResidue
BGLN241
BGLN244
BTHR245
BTYR248
BHOH701
BHOH764

site_idAC3
Number of Residues1
Detailsbinding site for residue PEG B 603
ChainResidue
BCEF601

site_idAC4
Number of Residues20
Detailsbinding site for residue CEF B 601
ChainResidue
BGLU307
BPRO308
BGLY309
BALA311
BILE312
BLYS313
BSER362
BASN364
BPHE420
BGLY421
BTYR422
BLYS497
BTHR498
BGLY499
BTHR500
BALA501
BARG502
BTYR544
BPEG603
BHOH771

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsACT_SITE: Acyl-ester intermediate => ECO:0000255|HAMAP-Rule:MF_02080
ChainResidueDetails
AGLY324
BGLY324

222415

PDB entries from 2024-07-10

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