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6P05

Bromodomain-containing protein 4 (BRD4) bromodomain 1 (BD1) complexed with compound 27

Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue GOL A 201
ChainResidue
AGLU49
AHOH393
AGLN62
ATYR118
AASN121
AALA122
AGLU167
AHOH315
AHOH331
AHOH342

site_idAC2
Number of Residues8
Detailsbinding site for residue GOL A 202
ChainResidue
ALEU42
AALA89
AVAL90
AASN93
ALEU94
APRO95
AASN162
AHOH366

site_idAC3
Number of Residues14
Detailsbinding site for residue YF2 A 203
ChainResidue
ATRP81
APRO82
APHE83
APRO86
AVAL87
AASP88
ALYS91
ALEU92
AASN140
AASP145
AHOH332
AHOH374
AHOH382
AHOH390

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99

218853

PDB entries from 2024-04-24

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