Loading
PDBj
MenuPDBj@FacebookPDBj@X(formerly Twitter)PDBj@BlueSkyPDBj@YouTubewwPDB FoundationwwPDBDonate
RCSB PDBPDBeBMRBAdv. SearchSearch help

6OWC

Mutant estrogen receptor alpha (ERa) Y537S covalently bound to H3B-6545.

Functional Information from PDB Data
site_idAC1
Number of Residues17
Detailsbinding site for residue ND1 A 601
ChainResidue
AMET343
ALEU391
APHE404
AILE424
ALEU428
AGLY521
ATYR526
ALYS529
ACYS530
ALEU346
ATHR347
AALA350
AASP351
AGLU353
ATRP383
ALEU387
AMET388

site_idAC2
Number of Residues8
Detailsbinding site for residue EDO B 602
ChainResidue
AARG434
AGLN506
ALEU509
AHOH735
BHIS476
BLEU479
BASP480
BHOH756

site_idAC3
Number of Residues19
Detailsbinding site for Di-peptide ND1 B 601 and CYS B 530
ChainResidue
BLEU346
BTHR347
BALA350
BGLU353
BLEU387
BMET388
BLEU391
BARG394
BPHE404
BMET421
BILE424
BPHE425
BLEU428
BGLY521
BLEU525
BMET528
BLYS529
BLYS531
BHOH730

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"9338790","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"9600906","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"1A52","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"1ERE","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues2
DetailsModified residue: {"description":"Phosphotyrosine; by Tyr-kinases","evidences":[{"source":"PubMed","id":"7539106","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues2
DetailsLipidation: {"description":"S-palmitoyl cysteine","evidences":[{"evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

239492

PDB entries from 2025-07-30

PDB statisticsPDBj update infoContact PDBjnumon