6OWC
Mutant estrogen receptor alpha (ERa) Y537S covalently bound to H3B-6545.
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 17 |
Details | binding site for residue ND1 A 601 |
Chain | Residue |
A | MET343 |
A | LEU391 |
A | PHE404 |
A | ILE424 |
A | LEU428 |
A | GLY521 |
A | TYR526 |
A | LYS529 |
A | CYS530 |
A | LEU346 |
A | THR347 |
A | ALA350 |
A | ASP351 |
A | GLU353 |
A | TRP383 |
A | LEU387 |
A | MET388 |
site_id | AC2 |
Number of Residues | 8 |
Details | binding site for residue EDO B 602 |
Chain | Residue |
A | ARG434 |
A | GLN506 |
A | LEU509 |
A | HOH735 |
B | HIS476 |
B | LEU479 |
B | ASP480 |
B | HOH756 |
site_id | AC3 |
Number of Residues | 19 |
Details | binding site for Di-peptide ND1 B 601 and CYS B 530 |
Chain | Residue |
B | LEU346 |
B | THR347 |
B | ALA350 |
B | GLU353 |
B | LEU387 |
B | MET388 |
B | LEU391 |
B | ARG394 |
B | PHE404 |
B | MET421 |
B | ILE424 |
B | PHE425 |
B | LEU428 |
B | GLY521 |
B | LEU525 |
B | MET528 |
B | LYS529 |
B | LYS531 |
B | HOH730 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 6 |
Details | Binding site: {"evidences":[{"source":"PubMed","id":"9338790","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"9600906","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"1A52","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"1ERE","evidenceCode":"ECO:0007744"}]} |
Chain | Residue | Details |
site_id | SWS_FT_FI2 |
Number of Residues | 2 |
Details | Modified residue: {"description":"Phosphotyrosine; by Tyr-kinases","evidences":[{"source":"PubMed","id":"7539106","evidenceCode":"ECO:0000269"}]} |
Chain | Residue | Details |
site_id | SWS_FT_FI3 |
Number of Residues | 2 |
Details | Lipidation: {"description":"S-palmitoyl cysteine","evidences":[{"evidenceCode":"ECO:0000250"}]} |
Chain | Residue | Details |