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6O9W

Crystal structure of Staphylococcus aureus BlaR1 antibiotic-sensor domain in complex with avibactam

Functional Information from GO Data
ChainGOidnamespacecontents
A0008658molecular_functionpenicillin binding
B0008658molecular_functionpenicillin binding
Functional Information from PDB Data
site_idAC1
Number of Residues18
Detailsbinding site for residue NXL A 601
ChainResidue
AASN388
AGLY528
ATHR529
AGLY530
AILE531
AHOH710
BILE531
BASN533
BGLY534
BNXL601
ASER389
ALYS392
ASER437
AASN439
AMET476
AGLU477
ALYS526
ATHR527

site_idAC2
Number of Residues19
Detailsbinding site for Di-peptide NXL B 601 and SER B 389
ChainResidue
AILE531
AGLY534
ANXL601
AHOH710
BPRO387
BASN388
BTHR390
BTYR391
BLYS392
BSER437
BASN439
BMET476
BGLU477
BLYS526
BTHR527
BGLY528
BTHR529
BGLY530
BILE531

site_idAC3
Number of Residues19
Detailsbinding site for Di-peptide NXL B 601 and SER B 389
ChainResidue
AILE531
AGLY534
ANXL601
AHOH710
BPRO387
BASN388
BTHR390
BTYR391
BLYS392
BSER437
BASN439
BMET476
BGLU477
BLYS526
BTHR527
BGLY528
BTHR529
BGLY530
BILE531

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsACT_SITE: Acyl-ester intermediate => ECO:0000269|PubMed:15506754, ECO:0000269|PubMed:21775440
ChainResidueDetails
ASER389
BSER389

site_idSWS_FT_FI2
Number of Residues2
DetailsMOD_RES: N6-carboxylysine => ECO:0000269|PubMed:12591921
ChainResidueDetails
ALYS392
BLYS392

223532

PDB entries from 2024-08-07

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