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6O4U

Co-crystal structure of Mcl1 with inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0042981biological_processregulation of apoptotic process
B0042981biological_processregulation of apoptotic process
Functional Information from PDB Data
site_idAC1
Number of Residues16
Detailsbinding site for residue LMV A 401
ChainResidue
APHE228
AHOH566
AHOH570
BHIS224
BPHE228
BTHR266
BLMV401
BHOH554
AMET231
AMET250
AVAL253
AARG263
ALEU267
APHE270
ALEU290
AHOH522

site_idAC2
Number of Residues12
Detailsbinding site for residue LMV B 401
ChainResidue
APHE228
ALMV401
AHOH566
BMET231
BVAL249
BMET250
BARG263
BLEU267
BPHE270
BGLY271
BHOH544
BHOH554

Functional Information from PROSITE/UniProt
site_idPS01080
Number of Residues20
DetailsBH1 Apoptosis regulator, Bcl-2 family BH1 motif signature. VFsDGvtNWGRIVTLIsFGA
ChainResidueDetails
AVAL253-ALA272

site_idPS01258
Number of Residues12
DetailsBH2 Apoptosis regulator, Bcl-2 family BH2 motif signature. WLvkqRGWDgFV
ChainResidueDetails
ATRP305-VAL316

site_idPS01259
Number of Residues15
DetailsBH3 Apoptosis regulator, Bcl-2 family BH3 motif signature. AletLRrVGDGVQRN
ChainResidueDetails
AALA209-ASN223

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues28
DetailsMotif: {"description":"BH3"}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues40
DetailsMotif: {"description":"BH1"}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues30
DetailsMotif: {"description":"BH2"}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues5
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin)"}
ChainResidueDetails

243911

PDB entries from 2025-10-29

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