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6NWK

Structure of the Ancestral Glucocorticoid Receptor 2 ligand binding domain in complex with dexamethasone and PGC1a coregulator fragment

Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue DEX A 301
ChainResidue
AMET29
ACYS205
ATHR208
AVAL216
ALEU32
AASN33
AGLY36
AGLN39
AARG80
APHE92
AGLN111
APHE204

site_idAC2
Number of Residues5
Detailsbinding site for residue FMT A 302
ChainResidue
APRO51
AGLN203
APHE206
ALYS234
AHOH407

site_idAC3
Number of Residues5
Detailsbinding site for residue ACE A 303
ChainResidue
AARG54
AASN55
AGLY200
APHE204
AHOH407

site_idAC4
Number of Residues5
Detailsbinding site for residue DMS A 304
ChainResidue
ATYR82
ALYS83
AASN86
AASN86
AASN88

site_idAC5
Number of Residues6
Detailsbinding site for residue DMS A 305
ChainResidue
AGLU9
AVAL12
ASER76
AARG80
ATYR132
AHOH421

site_idAC6
Number of Residues9
Detailsbinding site for residue GOL A 306
ChainResidue
AGLU9
APRO10
AALA43
ATRP46
ALEU72
AMET73
ASER76
ALYS136
AHOH446

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: N6-acetyllysine => ECO:0000250|UniProtKB:O70343
ChainResidueDetails
BLYS146

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PDB entries from 2024-09-11

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