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6L96

Structure of PPARalpha-LBD/pemafibrate/SRC1 peptide

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0005634cellular_componentnucleus
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues15
Detailsbinding site for residue P7F A 501
ChainResidue
AVAL256
ALEU321
AVAL324
AVAL332
AMET355
AHIS440
ATYR464
APHE273
ACYS275
ACYS276
ATHR279
ASER280
ATYR314
AILE317
APHE318

site_idAC2
Number of Residues17
Detailsbinding site for residue P7F B 501
ChainResidue
BLEU247
BPHE273
BCYS275
BCYS276
BTHR279
BSER280
BTYR314
BPHE318
BMET320
BLEU321
BVAL324
BMET330
BVAL332
BMET355
BHIS440
BLEU460
BTYR464

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues258
DetailsRegion: {"description":"Required for heterodimerization with RXRA"}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues6
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"19116277","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"3ET1","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues2
DetailsSite: {"description":"Essential for heterodimerization with RXRA"}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues4
DetailsMotif: {"description":"LXXLL motif 4"}
ChainResidueDetails

239492

PDB entries from 2025-07-30

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