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6L6K

Crystal structure of dimeric RXRalpha-LBD complexed with partial agonist CBt-PMN and SRC1

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0003707molecular_functionnuclear steroid receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
A0008270molecular_functionzinc ion binding
Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue 9HF A 501
ChainResidue
AILE268
AILE345
ACYS432
AHIS435
AHOH615
AALA271
AALA272
AGLN275
ALEU309
APHE313
AARG316
ALEU326
AALA327

site_idAC2
Number of Residues7
Detailsbinding site for residue CA A 502
ChainResidue
AGLU434
AGLU434
AHOH606
AHOH728
AHOH744
AHOH744
AHOH750

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163
ChainResidueDetails
BSER698
AALA327

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:24275569
ChainResidueDetails
ASER259

site_idSWS_FT_FI3
Number of Residues1
DetailsMOD_RES: Phosphoserine; by MAPK8 and MAPK9 => ECO:0000250|UniProtKB:P28700
ChainResidueDetails
ASER260

223532

PDB entries from 2024-08-07

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