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6KNU

THRb mutation with a novel agonist

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues15
Detailsbinding site for residue 8HO A 501
ChainResidue
APHE272
ALEU330
AASN331
AGLY344
ALEU346
AHOH601
AHOH621
AILE276
AALA279
AARG282
AMET310
AMET313
ASER314
AARG316
AALA317

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"15466465","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"1Y0X","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues4
DetailsMotif: {"description":"LXXLL motif 3"}
ChainResidueDetails

239803

PDB entries from 2025-08-06

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