Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

6KB8

X-ray structure of human PPARalpha ligand binding domain-GW7647 co-crystals obtained by cross-seeding

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue GOL A 501
ChainResidue
ALYS222
AARG226
ASER323
AMET325
AASN326
AASN366

site_idAC2
Number of Residues13
Detailsbinding site for residue 2VN A 502
ChainResidue
ATHR279
ASER280
ATHR283
ATYR314
AMET355
AHIS440
ALEU456
ATYR464
AHOH618
AHOH677
APHE273
ACYS276
AGLN277

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsBINDING: BINDING => ECO:0000269|PubMed:19116277, ECO:0007744|PDB:3ET1
ChainResidueDetails
ASER280
ATYR314
ATYR464

site_idSWS_FT_FI2
Number of Residues1
DetailsSITE: Essential for heterodimerization with RXRA
ChainResidueDetails
ALEU433

222926

PDB entries from 2024-07-24

PDB statisticsPDBj update infoContact PDBjnumon