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6J64

Crystal structure of human HINT1 mutant complexing with AP4A

Functional Information from GO Data
ChainGOidnamespacecontents
A0000118cellular_componenthistone deacetylase complex
A0000166molecular_functionnucleotide binding
A0003824molecular_functioncatalytic activity
A0005080molecular_functionprotein kinase C binding
A0005515molecular_functionprotein binding
A0005634cellular_componentnucleus
A0005654cellular_componentnucleoplasm
A0005737cellular_componentcytoplasm
A0005829cellular_componentcytosol
A0005856cellular_componentcytoskeleton
A0005886cellular_componentplasma membrane
A0006355biological_processregulation of DNA-templated transcription
A0006508biological_processproteolysis
A0006915biological_processapoptotic process
A0007165biological_processsignal transduction
A0008234molecular_functioncysteine-type peptidase activity
A0009154biological_processpurine ribonucleotide catabolic process
A0016787molecular_functionhydrolase activity
A0016926biological_processprotein desumoylation
A0016929molecular_functiondeSUMOylase activity
A0043530molecular_functionadenosine 5'-monophosphoramidase activity
A0050850biological_processpositive regulation of calcium-mediated signaling
A0070062cellular_componentextracellular exosome
A0072332biological_processintrinsic apoptotic signaling pathway by p53 class mediator
B0000118cellular_componenthistone deacetylase complex
B0000166molecular_functionnucleotide binding
B0003824molecular_functioncatalytic activity
B0005080molecular_functionprotein kinase C binding
B0005515molecular_functionprotein binding
B0005634cellular_componentnucleus
B0005654cellular_componentnucleoplasm
B0005737cellular_componentcytoplasm
B0005829cellular_componentcytosol
B0005856cellular_componentcytoskeleton
B0005886cellular_componentplasma membrane
B0006355biological_processregulation of DNA-templated transcription
B0006508biological_processproteolysis
B0006915biological_processapoptotic process
B0007165biological_processsignal transduction
B0008234molecular_functioncysteine-type peptidase activity
B0009154biological_processpurine ribonucleotide catabolic process
B0016787molecular_functionhydrolase activity
B0016926biological_processprotein desumoylation
B0016929molecular_functiondeSUMOylase activity
B0043530molecular_functionadenosine 5'-monophosphoramidase activity
B0050850biological_processpositive regulation of calcium-mediated signaling
B0070062cellular_componentextracellular exosome
B0072332biological_processintrinsic apoptotic signaling pathway by p53 class mediator
Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue TAU B 201
ChainResidue
BTHR17
BHOH344
BTHR17
BILE18
BILE18
BHOH320
BHOH320
BHOH328
BHOH328
BHOH344

site_idAC2
Number of Residues29
Detailsbinding site for residue B4P B 202
ChainResidue
BILE18
BILE18
BPHE19
BPRO28
BPHE41
BPHE41
BHIS42
BHIS42
BASP43
BILE44
BILE44
BSER45
BLEU53
BGLN106
BSER107
BVAL108
BHIS112
BHOH301
BHOH315
BHOH317
BHOH317
BHOH319
BHOH321
BHOH329
BHOH361
BHOH404
BHOH411
BHOH446
BHOH446

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsACT_SITE: Tele-AMP-histidine intermediate => ECO:0000269|PubMed:9323207
ChainResidueDetails
AHIS112
BHIS112

site_idSWS_FT_FI2
Number of Residues8
DetailsBINDING: BINDING => ECO:0000269|PubMed:22869114, ECO:0007744|PDB:3TW2
ChainResidueDetails
AASP43
AASN99
AGLY105
AHIS112
BASP43
BASN99
BGLY105
BHIS112

site_idSWS_FT_FI3
Number of Residues2
DetailsMOD_RES: N-acetylalanine => ECO:0007744|PubMed:22814378
ChainResidueDetails
AALA2
BALA2

site_idSWS_FT_FI4
Number of Residues4
DetailsMOD_RES: N6-acetyllysine => ECO:0007744|PubMed:19608861
ChainResidueDetails
ALYS21
ALYS30
BLYS21
BLYS30

site_idSWS_FT_FI5
Number of Residues4
DetailsMOD_RES: Phosphoserine => ECO:0000250|UniProtKB:P70349
ChainResidueDetails
ASER45
ASER72
BSER45
BSER72

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PDB entries from 2024-07-10

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