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6ITM

Crystal structure of FXR in complex with agonist XJ034

Functional Information from GO Data
ChainGOidnamespacecontents
A0004879molecular_functionnuclear receptor activity
A0032052molecular_functionbile acid binding
A0038183biological_processbile acid signaling pathway
C0004879molecular_functionnuclear receptor activity
C0032052molecular_functionbile acid binding
C0038183biological_processbile acid signaling pathway
Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue AWL A 501
ChainResidue
APHE298
AILE371
ATYR375
ATYR383
AMET464
ALEU301
ATHR302
AMET304
AHIS308
AMET342
ASER346
AILE349
ALEU362

site_idAC2
Number of Residues8
Detailsbinding site for residue AWL C 501
ChainResidue
CPHE298
CTHR302
CMET304
CHIS308
CSER346
CILE366
CTYR375
CTRP483

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsBinding site: {"evidences":[{"source":"PDB","id":"6HL1","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues2
DetailsModified residue: {"description":"Phosphothreonine; by PKC/PRKCZ","evidences":[{"source":"PubMed","id":"18668687","evidenceCode":"ECO:0000305"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues4
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO1)","evidences":[{"source":"PubMed","id":"23546875","evidenceCode":"ECO:0000305"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues8
DetailsMotif: {"description":"LXXLL motif 5"}
ChainResidueDetails

238582

PDB entries from 2025-07-09

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