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6IN1

Crystal structure of the first bromodomain of BRD4 in complex with 18-Crown-6

Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue LOC A 200
ChainResidue
APRO82
AHOH316
AHOH322
AHOH392
APHE83
AVAL87
ALEU94
AASP96
ALYS99
AASN140
AASP144
AILE146

site_idAC2
Number of Residues10
Detailsbinding site for residue O4B A 201
ChainResidue
ATYR65
AVAL69
ATHR73
ATHR134
ATYR137
AGLU151
AGLU154
ALEU156
ALYS160
AGLU163

site_idAC3
Number of Residues5
Detailsbinding site for residue NA A 202
ChainResidue
ATYR137
AILE138
AASN140
AGLU163
AHOH414

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99

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PDB entries from 2024-07-31

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