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6HJ2

Crystal structure of hPXR in complex with dabrafenib

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue P06 A 501
ChainResidue
AMET243
AMET425
APHE429
AHOH602
AHOH624
ASER247
APHE251
APHE281
ACYS284
AGLN285
ATRP299
AHIS407
ALEU411

site_idAC2
Number of Residues1
Detailsbinding site for residue IPA A 502
ChainResidue
ALEU276

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues5
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"12578355","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"1M13","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

238582

PDB entries from 2025-07-09

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