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6HDN

Crystal structure of human ATAD2 bromodomain in complex with 3-methyl-8-((8-methyl-8-azabicyclooctan-3-yl)amino)-1,7-naphthyridin-2(1H)-one

Functional Information from GO Data
ChainGOidnamespacecontents
A0006325biological_processchromatin organization
A0006355biological_processregulation of transcription, DNA-templated
A0016887molecular_functionATP hydrolysis activity
Functional Information from PDB Data
site_idAC1
Number of Residues5
Detailsbinding site for residue SO4 A 1201
ChainResidue
ALEU1073
AARG1077
AHOH1307
AHOH1341
AHOH1396

site_idAC2
Number of Residues8
Detailsbinding site for residue SO4 A 1202
ChainResidue
AARG1072
AHOH1303
AHOH1308
AHOH1423
AARG987
AARG990
AARG994
AARG1067

site_idAC3
Number of Residues5
Detailsbinding site for residue SO4 A 1203
ChainResidue
ALYS1037
ALYS1042
AHOH1361
AHOH1379
AHOH1379

site_idAC4
Number of Residues6
Detailsbinding site for residue EDO A 1204
ChainResidue
AHIS998
AGLU1091
AGLU1092
AASP1094
AHOH1372
AHOH1427

site_idAC5
Number of Residues6
Detailsbinding site for residue EDO A 1205
ChainResidue
AGLU988
ALEU1093
AASP1094
APHE1097
AHOH1326
AHOH1376

site_idAC6
Number of Residues7
Detailsbinding site for residue FZB A 1206
ChainResidue
AVAL1008
AVAL1013
AGLU1017
AASN1064
AASP1071
AILE1074
AHOH1310

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PDB entries from 2024-05-01

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