Functional Information from GO Data
Chain | GOid | namespace | contents |
A | 0004672 | molecular_function | protein kinase activity |
A | 0004713 | molecular_function | protein tyrosine kinase activity |
A | 0004714 | molecular_function | transmembrane receptor protein tyrosine kinase activity |
A | 0005524 | molecular_function | ATP binding |
A | 0006468 | biological_process | protein phosphorylation |
A | 0007169 | biological_process | cell surface receptor protein tyrosine kinase signaling pathway |
A | 0016020 | cellular_component | membrane |
B | 0004672 | molecular_function | protein kinase activity |
B | 0004713 | molecular_function | protein tyrosine kinase activity |
B | 0004714 | molecular_function | transmembrane receptor protein tyrosine kinase activity |
B | 0005524 | molecular_function | ATP binding |
B | 0006468 | biological_process | protein phosphorylation |
B | 0007169 | biological_process | cell surface receptor protein tyrosine kinase signaling pathway |
B | 0016020 | cellular_component | membrane |
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 20 |
Details | binding site for residue FEW A 1001 |
Chain | Residue |
A | VAL624 |
A | THR701 |
A | ASP702 |
A | TYR703 |
A | MET704 |
A | PHE762 |
A | HIS764 |
A | LEU773 |
A | ALA783 |
A | ASP784 |
A | EDO1012 |
A | ALA653 |
A | HOH1253 |
A | LYS655 |
A | GLU672 |
A | ILE675 |
A | MET676 |
A | LEU679 |
A | ILE685 |
A | MET699 |
site_id | AC2 |
Number of Residues | 5 |
Details | binding site for residue SO4 A 1002 |
Chain | Residue |
A | SER788 |
A | ARG789 |
A | ASN790 |
A | LEU791 |
A | HOH1165 |
site_id | AC3 |
Number of Residues | 7 |
Details | binding site for residue SO4 A 1003 |
Chain | Residue |
A | HIS745 |
A | ALA748 |
A | GLN749 |
A | SER752 |
A | HIS902 |
A | ALA906 |
A | HOH1164 |
site_id | AC4 |
Number of Residues | 4 |
Details | binding site for residue SO4 A 1004 |
Chain | Residue |
A | ARG755 |
A | ARG903 |
A | HOH1124 |
A | HOH1171 |
site_id | AC5 |
Number of Residues | 6 |
Details | binding site for residue SO4 A 1005 |
Chain | Residue |
A | ARG872 |
A | PRO874 |
A | ALA875 |
B | GLY801 |
B | ARG802 |
B | ARG903 |
site_id | AC6 |
Number of Residues | 8 |
Details | binding site for residue EDO A 1006 |
Chain | Residue |
A | TRP834 |
A | PHE845 |
A | GLY846 |
A | LEU870 |
A | SER871 |
A | EDO1013 |
A | HOH1184 |
B | LYS671 |
site_id | AC7 |
Number of Residues | 6 |
Details | binding site for residue EDO A 1007 |
Chain | Residue |
A | TRP827 |
A | PHE845 |
A | TYR869 |
A | LEU870 |
A | TRP888 |
A | HOH1151 |
site_id | AC8 |
Number of Residues | 5 |
Details | binding site for residue EDO A 1008 |
Chain | Residue |
A | ARG866 |
A | HOH1143 |
A | HOH1172 |
B | LEU670 |
B | LYS674 |
site_id | AC9 |
Number of Residues | 6 |
Details | binding site for residue EDO A 1009 |
Chain | Residue |
A | ARG678 |
A | LEU760 |
A | ASN761 |
B | GLY846 |
B | LEU848 |
B | EDO1007 |
site_id | AD1 |
Number of Residues | 5 |
Details | binding site for residue EDO A 1010 |
Chain | Residue |
A | LEU670 |
A | VAL673 |
A | LYS674 |
B | ARG866 |
B | EDO1005 |
site_id | AD2 |
Number of Residues | 1 |
Details | binding site for residue EDO A 1011 |
site_id | AD3 |
Number of Residues | 1 |
Details | binding site for residue EDO A 1012 |
site_id | AD4 |
Number of Residues | 4 |
Details | binding site for residue EDO A 1013 |
Chain | Residue |
A | TRP834 |
A | MET838 |
A | EDO1006 |
A | HOH1184 |
site_id | AD5 |
Number of Residues | 2 |
Details | binding site for residue EDO A 1014 |
Chain | Residue |
A | ALA875 |
A | PRO877 |
site_id | AD6 |
Number of Residues | 5 |
Details | binding site for residue EDO A 1015 |
Chain | Residue |
A | MET787 |
A | ALA793 |
A | TYR796 |
A | ARG798 |
A | GLU907 |
site_id | AD7 |
Number of Residues | 17 |
Details | binding site for residue FEW B 1001 |
Chain | Residue |
B | ALA783 |
B | ASP784 |
B | HOH1191 |
B | VAL624 |
B | ALA653 |
B | LYS655 |
B | GLU672 |
B | MET676 |
B | LEU679 |
B | MET699 |
B | THR701 |
B | ASP702 |
B | TYR703 |
B | MET704 |
B | PHE762 |
B | HIS764 |
B | LEU773 |
site_id | AD8 |
Number of Residues | 6 |
Details | binding site for residue SO4 B 1002 |
Chain | Residue |
A | GLY801 |
A | ARG802 |
A | ARG903 |
B | ARG872 |
B | PRO874 |
B | ALA875 |
site_id | AD9 |
Number of Residues | 6 |
Details | binding site for residue SO4 B 1003 |
Chain | Residue |
A | LYS671 |
B | TRP834 |
B | PHE845 |
B | LEU870 |
B | SER871 |
B | HOH1197 |
site_id | AE1 |
Number of Residues | 6 |
Details | binding site for residue EDO B 1004 |
Chain | Residue |
B | TRP827 |
B | PHE845 |
B | TYR869 |
B | LEU870 |
B | TRP888 |
B | HOH1152 |
site_id | AE2 |
Number of Residues | 6 |
Details | binding site for residue EDO B 1005 |
Chain | Residue |
A | MET600 |
A | LYS674 |
A | EDO1010 |
B | GLU855 |
B | GLU859 |
B | ARG866 |
site_id | AE3 |
Number of Residues | 5 |
Details | binding site for residue EDO B 1006 |
Chain | Residue |
B | MET787 |
B | ALA793 |
B | TYR796 |
B | ARG798 |
B | HOH1112 |
site_id | AE4 |
Number of Residues | 7 |
Details | binding site for residue EDO B 1007 |
Chain | Residue |
A | EDO1009 |
B | GLY794 |
B | ARG808 |
B | GLN843 |
B | ASP850 |
B | HOH1139 |
B | HOH1140 |
site_id | AE5 |
Number of Residues | 3 |
Details | binding site for residue EDO B 1008 |
Chain | Residue |
A | MET838 |
B | GLN800 |
B | ALA803 |
Functional Information from PROSITE/UniProt
site_id | PS00109 |
Number of Residues | 13 |
Details | PROTEIN_KINASE_TYR Tyrosine protein kinases specific active-site signature. FVHrDLATRNCLV |
Chain | Residue | Details |
A | PHE762-VAL774 | |
site_id | PS00239 |
Number of Residues | 9 |
Details | RECEPTOR_TYR_KIN_II Receptor tyrosine kinase class II signature. NLYagdYYR |
Chain | Residue | Details |
A | ASN790-ARG798 | |
Functional Information from SwissProt/UniProt
Chain | Residue | Details |
A | PHE785 | |
B | PHE785 | |
Chain | Residue | Details |
A | LEU635 | |
B | LEU635 | |
site_id | SWS_FT_FI3 |
Number of Residues | 2 |
Details | BINDING: |
Chain | Residue | Details |
A | LYS674 | |
B | LYS674 | |
Chain | Residue | Details |
A | LEU650 | |
B | LEU650 | |
Chain | Residue | Details |
A | THR759 | |
B | THR759 | |
Chain | Residue | Details |
A | ALA811 | |
A | ILE815 | |
A | LEU816 | |
B | ALA811 | |
B | ILE815 | |
B | LEU816 | |