Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

6GRO

Human CSNK1G3 bound to SB-223133

Functional Information from GO Data
ChainGOidnamespacecontents
A0004672molecular_functionprotein kinase activity
A0004674molecular_functionprotein serine/threonine kinase activity
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
Functional Information from PDB Data
site_idAC1
Number of Residues7
Detailsbinding site for residue EDO A 401
ChainResidue
AARG161
AASP162
AVAL163
ATHR212
AMET216
AALA234
AHOH581

site_idAC2
Number of Residues4
Detailsbinding site for residue EDO A 402
ChainResidue
ATYR152
AHOH790
AASN66
ASER148

site_idAC3
Number of Residues1
Detailsbinding site for residue CL A 403
ChainResidue
AARG44

site_idAC4
Number of Residues5
Detailsbinding site for residue EDO A 404
ChainResidue
ASER208
ATHR210
ATHR220
AGLN226
AHOH560

site_idAC5
Number of Residues6
Detailsbinding site for residue EDO A 405
ChainResidue
APHE43
AASN62
ATHR65
AGLU67
AVAL69
ATYR103

site_idAC6
Number of Residues16
Detailsbinding site for residue F92 A 406
ChainResidue
ALEU57
AALA70
ALYS72
AMET114
ALEU116
AGLU117
ALEU118
ALEU119
AASP125
AGLU166
AILE184
AHOH511
AHOH580
AHOH594
AHOH612
AHOH737

Functional Information from PROSITE/UniProt
site_idPS00107
Number of Residues24
DetailsPROTEIN_KINASE_ATP Protein kinases ATP-binding region signature. IGCGNFGELRlGknlytney..........VAIK
ChainResidueDetails
AILE49-LYS72

site_idPS00108
Number of Residues13
DetailsPROTEIN_KINASE_ST Serine/Threonine protein kinases active-site signature. LiYrDVKpeNFLI
ChainResidueDetails
ALEU158-ILE170

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsACT_SITE: Proton acceptor => ECO:0000255|PROSITE-ProRule:PRU00159, ECO:0000255|PROSITE-ProRule:PRU10027
ChainResidueDetails
AASP162

site_idSWS_FT_FI2
Number of Residues2
DetailsBINDING: BINDING => ECO:0000255|PROSITE-ProRule:PRU00159
ChainResidueDetails
AILE49
ALYS72

226262

PDB entries from 2024-10-16

PDB statisticsPDBj update infoContact PDBjnumon