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6GGN

In vitro and in vivo characterization of a novel, highly potent p53-MDM2 inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0005634cellular_componentnucleus
A0043066biological_processnegative regulation of apoptotic process
A0051726biological_processregulation of cell cycle
Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue EYH A 201
ChainResidue
ALEU54
AGLY58
ATYR67
AGLN72
AVAL93
AHIS96
AILE99
ATYR100
AHOH319

site_idAC2
Number of Residues8
Detailsbinding site for residue CL A 202
ChainResidue
ATYR60
ALYS64
ALYS64
AASP80
AASP80
ALEU81
ALEU81
AHOH324

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues83
DetailsDomain: {"description":"SWIB/MDM2","evidences":[{"source":"PROSITE-ProRule","id":"PRU01273","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

247536

PDB entries from 2026-01-14

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