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6FZM

Human PARP14 (ARTD8), catalytic fragment in complex with inhibitor ITK6

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+ poly-ADP-ribosyltransferase activity
B0003950molecular_functionNAD+ poly-ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues11
Detailsbinding site for residue EE5 A 1901
ChainResidue
AHIS1682
ATYR1727
BHIS1779
AGLY1683
ALYS1704
AASN1705
AALA1706
ATYR1714
ATYR1721
ASER1722
ATHR1726

site_idAC2
Number of Residues8
Detailsbinding site for residue EE5 B 1901
ChainResidue
BHIS1682
BGLY1683
BTYR1701
BTYR1714
BTYR1721
BSER1722
BTHR1726
BTYR1727

240971

PDB entries from 2025-08-27

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