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6FR0

Crystal structure of CREBBP bromodomain complexd with PB08

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0006355biological_processregulation of DNA-templated transcription
B0004402molecular_functionhistone acetyltransferase activity
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue E3H A 1201
ChainResidue
APRO1110
AHOH1361
AHOH1366
BTRP1158
BTRP1165
AGLN1113
AVAL1115
ALEU1120
AILE1122
AASN1168
AARG1173
AHOH1306
AHOH1352

site_idAC2
Number of Residues10
Detailsbinding site for residue E3H B 1201
ChainResidue
ATRP1158
BPRO1110
BGLN1113
BVAL1115
BLEU1120
BASN1168
BARG1173
BHOH1306
BHOH1364
BHOH1369

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. SlpFrqpvDpqllgipDYFdiVknpMdlstIkrkldtgq..Yqepwqyvddvwl.MfnNAwlY
ChainResidueDetails
ASER1108-TYR1167

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PDB entries from 2024-04-24

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