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6FIC

Bivalent Inhibitor UNC4512 Bound to the TAF1 Bromodomain Tandem

Functional Information from GO Data
ChainGOidnamespacecontents
T0004402molecular_functionhistone acetyltransferase activity
T0005669cellular_componenttranscription factor TFIID complex
T0006366biological_processtranscription by RNA polymerase II
T0016251molecular_functionRNA polymerase II general transcription initiation factor activity
T0017025molecular_functionTBP-class protein binding
Functional Information from PDB Data
site_idAC1
Number of Residues14
Detailsbinding site for residue DKH T 1701
ChainResidue
TPRO1404
TALA1577
TVAL1580
THOH1802
THOH1806
THOH1867
TTHR1407
TPRO1408
TVAL1409
TASN1410
TVAL1414
TASN1460
THIS1464
TLEU1466

site_idAC2
Number of Residues11
Detailsbinding site for residue DKH T 1702
ChainResidue
TTRP1526
TPRO1527
TPRO1527
TPHE1528
TPRO1531
TASN1533
TVAL1537
TASN1583
TTYR1589
TTYR1589
THOH1825

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. TypFhtpvNakvvk..DYYkiItrpMdlqtLrenvrkrl..Ypsreefrehlel.IvkNSatY
ChainResidueDetails
TTHR1402-TYR1459
TSER1525-TYR1582

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues109
DetailsDomain: {"description":"Bromo 2","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

248335

PDB entries from 2026-01-28

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