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6FFE

Human BRD2 C-terminal bromodomain with 2-((4-acetyl-3-cyclopropyl-3,4-dihydroquinoxalin-1(2H)-yl)methyl)benzoic acid

Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue PEG A 501
ChainResidue
ASER347
ALYS351
APEG502
AHOH601
AHOH621
AHOH671

site_idAC2
Number of Residues6
Detailsbinding site for residue PEG A 502
ChainResidue
APRO430
APEG501
AHOH621
ALYS351
AASP385
ATYR428

site_idAC3
Number of Residues6
Detailsbinding site for residue EDO A 503
ChainResidue
ATYR426
AARG440
AGLN443
AASP444
APHE448
AHOH619

site_idAC4
Number of Residues8
Detailsbinding site for residue EDO A 504
ChainResidue
ATYR368
ALYS402
AASP407
AGLU413
AMET438
ALYS441
AHOH603
AHOH654

site_idAC5
Number of Residues10
Detailsbinding site for residue D7Q A 505
ChainResidue
ATRP370
APRO371
ALEU383
ACYS425
ATYR428
AASN429
AVAL435
AMET438
AHOH617
AHOH691

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFykpvDasalglhDYHdiIkhpMdlstVkrkmenrd..Yrdaqefaadvrl.MfsNCykY
ChainResidueDetails
AALA369-TYR428

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues109
DetailsDomain: {"description":"Bromo 2","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

245663

PDB entries from 2025-12-03

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