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6EPW

The ATAD2 bromodomain in complex with compound UZH-DU32

Functional Information from GO Data
ChainGOidnamespacecontents
A0006325biological_processchromatin organization
A0006355biological_processregulation of transcription, DNA-templated
A0016887molecular_functionATP hydrolysis activity
Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue BQ8 A 1201
ChainResidue
AVAL1008
AVAL1013
ATYR1063
AASN1064
AGLY1070
AASP1071
AHOH1303
AHOH1317
AHOH1329

site_idAC2
Number of Residues10
Detailsbinding site for residue BQ8 A 1202
ChainResidue
APRO1012
AVAL1013
AASP1014
APRO1015
ATYR1021
AILE1025
APRO1028
AHOH1301
AHOH1301
AHOH1302

site_idAC3
Number of Residues4
Detailsbinding site for residue SO4 A 1203
ChainResidue
AARG987
AARG990
AARG994
AARG1067

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PDB entries from 2024-07-10

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