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6ENX

Zebrafish Sirt5 in complex with stalled bicyclic intermediate of inhibitory compound 10

Functional Information from GO Data
ChainGOidnamespacecontents
A0036054molecular_functionprotein-malonyllysine demalonylase activity
A0036055molecular_functionprotein-succinyllysine desuccinylase activity
A0070403molecular_functionNAD+ binding
Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue ZN A 301
ChainResidue
ACYS162
ACYS165
ACYS203
ACYS208

site_idAC2
Number of Residues7
Detailsbinding site for residue DMS A 302
ChainResidue
ABJW303
AHOH457
ATYR251
AALA254
APRO276
AALA277
AARG280

site_idAC3
Number of Residues39
Detailsbinding site for residue BJW A 303
ChainResidue
AGLY54
AALA55
AGLY56
ATHR65
APHE66
AARG67
ATRP73
ATYR98
AARG101
AGLN136
AILE138
AHIS154
AVAL217
ATRP218
APHE219
AGLY220
AGLU221
AGLU232
AGLY245
ATHR246
ASER247
AILE249
AVAL250
ATYR251
ATYR251
AMET255
APHE256
AGLN259
AASN271
AMET272
AGLU273
APRO288
ACYS289
ADMS302
AHOH404
AHOH415
AHOH416
AHOH443
AHOH452

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsACT_SITE: Proton acceptor => ECO:0000255|PROSITE-ProRule:PRU00236
ChainResidueDetails
AHIS154

site_idSWS_FT_FI2
Number of Residues11
DetailsBINDING: BINDING => ECO:0000255|HAMAP-Rule:MF_03160
ChainResidueDetails
ATYR98
AARG101
AGLN136
ACYS162
ACYS165
ACYS203
ACYS208
AGLY245
AASN271
ACYS289
AGLY54

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PDB entries from 2024-05-15

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