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6EL9

Glucocorticoid Receptor in complex with AZD9567

Functional Information from PDB Data
site_idAC1
Number of Residues5
Detailsbinding site for residue EDO A 801
ChainResidue
APRO541
AMET604
AALA607
ALYS667
AHOH934

site_idAC2
Number of Residues18
Detailsbinding site for residue B9W A 802
ChainResidue
AGLN570
ATRP600
AMET604
AALA607
AARG611
ACYS622
APHE623
AGLN642
AMET646
ACYS736
ATHR739
APHE749
ALEU753
AHOH934
ALEU563
AASN564
ALEU566
AGLY567

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues165
DetailsRegion: {"description":"Interaction with CRY1","evidences":[{"source":"PubMed","id":"22170608","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues2
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO)","evidences":[{"source":"PubMed","id":"12144530","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues4
DetailsMotif: {"description":"LXXLL motif 3"}
ChainResidueDetails

247536

PDB entries from 2026-01-14

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