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6E5V

human mGlu8 receptor amino terminal domain in complex with (S)-3,4-Dicarboxyphenylglycine (DCPG)

Functional Information from GO Data
ChainGOidnamespacecontents
A0004930molecular_functionG protein-coupled receptor activity
A0007186biological_processG protein-coupled receptor signaling pathway
A0016020cellular_componentmembrane
B0004930molecular_functionG protein-coupled receptor activity
B0007186biological_processG protein-coupled receptor signaling pathway
B0016020cellular_componentmembrane
Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue HVG A 601
ChainResidue
ALYS71
ASER310
ALYS314
ALYS401
AARG75
AALA154
AALA155
ASER156
AALA177
ATHR179
ATYR227
AASP309

site_idAC2
Number of Residues4
Detailsbinding site for residue CL A 602
ChainResidue
ATHR105
AALA154
AALA155
AVAL158

site_idAC3
Number of Residues12
Detailsbinding site for residue HVG B 601
ChainResidue
BLYS71
BARG75
BALA154
BSER156
BALA177
BSER178
BTHR179
BTYR227
BASP309
BSER310
BLYS314
BLYS401

site_idAC4
Number of Residues4
Detailsbinding site for residue CL B 602
ChainResidue
BTHR105
BALA154
BALA155
BVAL158

Functional Information from PROSITE/UniProt
site_idPS00979
Number of Residues19
DetailsG_PROTEIN_RECEP_F3_1 G-protein coupled receptors family 3 signature 1. VaNILrLFkIPQISyASTA
ChainResidueDetails
AVAL162-ALA180

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues10
DetailsBINDING: BINDING => ECO:0000250
ChainResidueDetails
ASER157
BVAL402
ASER178
AGLY228
ASER310
AVAL402
BSER157
BSER178
BGLY228
BSER310

site_idSWS_FT_FI2
Number of Residues8
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000255
ChainResidueDetails
AILE96
AGLN299
AGLY453
ALYS481
BILE96
BGLN299
BGLY453
BLYS481

222036

PDB entries from 2024-07-03

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