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6DVR

Crystal structure of human CARM1 with (R)-SKI-72

Functional Information from GO Data
ChainGOidnamespacecontents
A0016274molecular_functionprotein-arginine N-methyltransferase activity
A0018216biological_processpeptidyl-arginine methylation
B0016274molecular_functionprotein-arginine N-methyltransferase activity
B0018216biological_processpeptidyl-arginine methylation
Functional Information from PDB Data
site_idAC1
Number of Residues26
Detailsbinding site for residue HDG A 501
ChainResidue
ATYR149
AGLY192
ALEU198
AGLU214
AALA215
AGLY240
ALYS241
AVAL242
AGLU243
AGLU257
AMET259
APHE150
AGLU266
AMET268
ASER271
AP15502
AHOH624
AHOH657
AHOH740
APHE152
ATYR153
AGLN158
AGLN159
AASN161
AARG168
ATHR169

site_idAC2
Number of Residues8
Detailsbinding site for residue P15 A 502
ChainResidue
AASN161
AARG168
ATYR261
AHIS414
ATRP415
AHDG501
AHOH631
AHOH666

site_idAC3
Number of Residues25
Detailsbinding site for residue HDG B 501
ChainResidue
BTYR149
BPHE150
BPHE152
BTYR153
BGLN158
BGLN159
BASN161
BARG168
BGLY192
BLEU198
BGLU214
BALA215
BGLY240
BLYS241
BVAL242
BGLU243
BGLU257
BMET259
BGLU266
BMET268
BSER271
BP15502
BHOH616
BHOH694
BHOH699

site_idAC4
Number of Residues7
Detailsbinding site for residue P15 B 502
ChainResidue
BASN161
BARG168
BTYR261
BHIS414
BTRP415
BHDG501
BHOH707

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues66
DetailsRegion: {"description":"Required for nuclear translocation","evidences":[{"source":"UniProtKB","id":"Q9WVG6","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues12
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"21410432","evidenceCode":"ECO:0000305"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues2
DetailsModified residue: {"description":"Phosphoserine","evidences":[{"source":"PubMed","id":"19843527","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues4
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin)","evidences":[{"source":"PubMed","id":"34480022","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

246031

PDB entries from 2025-12-10

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