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6DNE

Crystal structure of human Bromodomain-containing protein 4 (BRD4) bromodomain with MS660

Functional Information from PDB Data
site_idAC1
Number of Residues20
Detailsbinding site for residue H1V A 501
ChainResidue
AASN54
BTRP81
BPRO82
BGLN85
BVAL87
BLEU92
BASN93
BLEU94
BASN140
BASP145
BILE146
ATRP81
BHOH501
APRO82
ALEU92
AASN93
ALEU94
AASN140
AASP145
AILE146

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140
AASN433
BASN140
BASN433

site_idSWS_FT_FI2
Number of Residues2
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:18669648, ECO:0007744|PubMed:24275569
ChainResidueDetails
ASER470
BSER470

site_idSWS_FT_FI3
Number of Residues4
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99
BLYS99

222415

PDB entries from 2024-07-10

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