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6D2I

JAK2 Pseudokinase V617F in complex with AT9283

Functional Information from GO Data
ChainGOidnamespacecontents
A0004672molecular_functionprotein kinase activity
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
B0004672molecular_functionprotein kinase activity
B0005524molecular_functionATP binding
B0006468biological_processprotein phosphorylation
Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue 35R A 901
ChainResidue
ALEU551
ASER633
ALEU680
ASER698
AILE559
ALEU579
ALYS581
AGLU627
APHE628
AVAL629
ALYS630
APHE631

site_idAC2
Number of Residues12
Detailsbinding site for residue 35R B 901
ChainResidue
BILE559
BLEU579
BLYS581
BGLU627
BVAL629
BLYS630
BPHE631
BGLY632
BSER633
BLYS677
BLEU680
BSER698

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsSite: {"description":"Breakpoint for translocation to form PCM1-JAK2 fusion protein"}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues2
DetailsModified residue: {"description":"Phosphotyrosine","evidences":[{"source":"PubMed","id":"23186163","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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