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6CN5

HUMAN RETENOID-RELATED ORPHAN RECEPTOR-GAMMA LIGAND- BINDING DOMAIN IN COMPLEX WITH INDOLE LIGAND CP9b IN INVERSE AGONIST CONFORMATION

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0005634cellular_componentnucleus
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues21
Detailsbinding site for residue F7M A 601
ChainResidue
ACYS285
AVAL376
APHE377
APHE388
ACYS393
ALEU396
AILE397
AILE400
APHE401
ASER404
AHIS479
AGLN286
AARG482
AHOH726
ALEU287
ACYS320
AHIS323
ALEU324
AMET365
AARG367
AALA368

site_idAC2
Number of Residues20
Detailsbinding site for residue F7M B 601
ChainResidue
BCYS285
BGLN286
BLEU287
BCYS320
BHIS323
BLEU324
BMET365
BARG367
BALA368
BVAL376
BPHE377
BPHE388
BCYS393
BLEU396
BILE400
BPHE401
BSER404
BHIS479
BHOH736
BHOH740

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PDB entries from 2024-06-26

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