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6CHW

Estrogen Receptor Alpha Y537S covalently bound to antagonist H3B-5942.

Functional Information from PDB Data
site_idAC1
Number of Residues14
Detailsbinding site for residue F3D A 601
ChainResidue
ALEU346
ALYS529
ACYS530
AEDO603
AHOH710
AHOH748
ATHR347
AALA350
AGLU353
ALEU387
AARG394
AGLY521
ALEU525
AMET528

site_idAC2
Number of Residues8
Detailsbinding site for residue EDO A 602
ChainResidue
ASER381
AALA382
ATRP383
ALEU384
AGLU385
ASER518
AMET522
AHOH751

site_idAC3
Number of Residues5
Detailsbinding site for residue EDO A 603
ChainResidue
AALA350
AASP351
ATRP383
AF3D601
AHOH758

site_idAC4
Number of Residues2
Detailsbinding site for residue EDO A 604
ChainResidue
AGLU323
ATRP393

site_idAC5
Number of Residues6
Detailsbinding site for residue DMS A 605
ChainResidue
AHIS476
ALEU479
AASP480
AGLN506
ALEU509
AHOH717

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: Phosphotyrosine; by Tyr-kinases => ECO:0000269|PubMed:7539106
ChainResidueDetails
ASER537

site_idSWS_FT_FI2
Number of Residues1
DetailsLIPID: S-palmitoyl cysteine => ECO:0000250
ChainResidueDetails
ACYS447

218853

PDB entries from 2024-04-24

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