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6C7A

Conformational Changes in a Class A Beta lactamase that Prime it for Catalysis

Functional Information from GO Data
ChainGOidnamespacecontents
A0008800molecular_functionbeta-lactamase activity
A0016787molecular_functionhydrolase activity
A0017001biological_processantibiotic catabolic process
A0030655biological_processbeta-lactam antibiotic catabolic process
A0046677biological_processresponse to antibiotic
Functional Information from PDB Data
site_idAC1
Number of Residues14
Detailsbinding site for residue SO4 A 301
ChainResidue
AALA69
AHOH532
AHOH544
AHOH600
AHOH649
AHOH736
ASER129
ALYS233
ATHR234
AGLY235
ASER236
ASO4302
AHOH459
AHOH466

site_idAC2
Number of Residues10
Detailsbinding site for residue SO4 A 302
ChainResidue
AALA69
ASER129
ATHR234
AGLY235
ASER236
ASO4301
AHOH459
AHOH466
AHOH532
AHOH649

site_idAC3
Number of Residues14
Detailsbinding site for residue SO4 A 303
ChainResidue
ALYS81
AALA197
AASN271
AASN273
AASP274
AHOH481
AHOH492
AHOH529
AHOH580
AHOH580
AHOH614
AHOH643
AHOH709
AHOH790

site_idAC4
Number of Residues6
Detailsbinding site for residue SO4 A 304
ChainResidue
AALA52
AARG177
AHOH412
AHOH530
AHOH554
AHOH659

site_idAC5
Number of Residues10
Detailsbinding site for residue SO4 A 305
ChainResidue
ATRP228
APRO250
AGLU251
AASN252
AHIS253
APHE287
AHOH479
AHOH490
AHOH651
AHOH671

site_idAC6
Number of Residues8
Detailsbinding site for residue SO4 A 306
ChainResidue
ALYS196
AGLU266
AGLN267
AHOH424
AHOH441
AHOH494
AHOH543
AHOH550

site_idAC7
Number of Residues6
Detailsbinding site for residue SO4 A 307
ChainResidue
ALYS87
AHIS88
AASN91
AHOH427
AHOH484
AHOH609

site_idAC8
Number of Residues7
Detailsbinding site for residue SO4 A 308
ChainResidue
AHIS88
AARG93
AHOH454
AHOH488
AHOH535
AHOH548
AHOH688

site_idAC9
Number of Residues3
Detailsbinding site for residue SO4 A 309
ChainResidue
ASER28
AVAL29
AHOH420

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsACT_SITE: Acyl-ester intermediate
ChainResidueDetails
AALA69

site_idSWS_FT_FI2
Number of Residues1
DetailsBINDING:
ChainResidueDetails
ALYS233

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PDB entries from 2024-07-24

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