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6C5Q

PPARg LBD bound to SR10171

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue EKS A 501
ChainResidue
AGLY284
AILE341
ASER342
ATYR473
AEKS502
ACSO285
APHE287
AARG288
ASER289
AILE326
AMET329
ALEU330
ALEU333

site_idAC2
Number of Residues13
Detailsbinding site for residue EKS A 502
ChainResidue
AGLY258
AGLU259
AILE262
APHE264
ALYS265
AHIS266
AILE279
AARG280
AGLN283
AMET348
ALEU465
ATYR473
AEKS501

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"9744270","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"2PRG","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues2
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin)","evidences":[{"source":"PubMed","id":"36737649","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

240971

PDB entries from 2025-08-27

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