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6B31

Structure of RORgt in complex with a novel inverse agonist 2

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0005634cellular_componentnucleus
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue CFJ A 600
ChainResidue
ACYS320
AHIS323
AVAL361
AMET365
AALA368
APHE377
APHE378
AHIS479
AHOH702

site_idAC2
Number of Residues9
Detailsbinding site for residue CFJ B 600
ChainResidue
BCYS320
BHIS323
BVAL361
BMET365
BALA368
BPHE377
BPHE378
BHOH701
BHOH703

223532

PDB entries from 2024-08-07

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