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6AU3

Crystal structure of SETDB1 Tudor domain with aryl triazole fragments

Functional Information from PDB Data
site_idAC1
Number of Residues7
Detailsbinding site for residue BWM A 501
ChainResidue
AGLY300
APHE332
ATRP387
AILE388
ATYR389
ASER392
AARG394

site_idAC2
Number of Residues5
Detailsbinding site for residue SO4 A 502
ChainResidue
ALYS364
AASP381
AHOH627
AARG209
ATRP363

site_idAC3
Number of Residues6
Detailsbinding site for residue SO4 A 503
ChainResidue
ALEU242
ASER243
AHIS246
AHOH608
AHOH617
AHOH626

site_idAC4
Number of Residues5
Detailsbinding site for residue SO4 A 504
ChainResidue
AHIS214
ALYS215
AHOH609
AHOH622
AHOH671

site_idAC5
Number of Residues4
Detailsbinding site for residue SO4 A 505
ChainResidue
AARG203
ALYS215
AASP250
ALYS383

site_idAC6
Number of Residues6
Detailsbinding site for residue EDO A 506
ChainResidue
ATYR193
ASER262
ATHR320
AHOH602
AHOH632
AHOH658

222036

PDB entries from 2024-07-03

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