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6ALC

CREBBP bromodomain in complex with Cpd 4 (1-(1-(cyclopropylmethyl)-3-(1H-indol-4-yl)-1,4,6,7-tetrahydro-5H-pyrazolo[4,3-c]pyridin-5-yl)ethan-1-one)

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0006355biological_processregulation of DNA-templated transcription
B0004402molecular_functionhistone acetyltransferase activity
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue DMS A 1201
ChainResidue
AVAL1115
AASN1168
AVAL1174
AHOH1308

site_idAC2
Number of Residues5
Detailsbinding site for residue EDO A 1202
ChainResidue
APRO1123
AASP1124
AARG1169
ASER1172
AHOH1356

site_idAC3
Number of Residues12
Detailsbinding site for residue BKD B 1201
ChainResidue
ATYR1102
ALEU1109
AARG1112
AHOH1340
BLEU1109
BPRO1110
BVAL1115
BILE1122
BASN1168
BVAL1174
BHOH1306
BHOH1344

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. SlpFrqpvDpqllgipDYFdiVknpMdlstIkrkldtgq..Yqepwqyvddvwl.MfnNAwlY
ChainResidueDetails
ASER1108-TYR1167

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PDB entries from 2024-07-31

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