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6AJX

Crystal structure of BRD4 in complex with isoliquiritigenin in the absence of DMSO

Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue HCC A 201
ChainResidue
APRO82
AASN140
AHOH302
AHOH308
AVAL87
ALEU92
ALEU94
AASP96
ATYR97
ALYS99
AILE100
ACYS136

site_idAC2
Number of Residues4
Detailsbinding site for residue NA A 202
ChainResidue
ATYR137
AILE138
AASN140
AGLU163

site_idAC3
Number of Residues3
Detailsbinding site for residue NA A 203
ChainResidue
ATYR65
ALYS160
AGLU163

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues106
DetailsDomain: {"description":"Bromo 1","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues1
DetailsSite: {"description":"Acetylated histone binding","evidences":[{"source":"PubMed","id":"22464331","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues2
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2)","evidences":[{"source":"PubMed","id":"28112733","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

238895

PDB entries from 2025-07-16

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