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6A84

Tankyrase-2 in complex with compound 15d

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+ ADP-ribosyltransferase activity
B0003950molecular_functionNAD+ ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue ZN A 1201
ChainResidue
ACYS1081
AHIS1084
ACYS1089
ACYS1092

site_idAC2
Number of Residues15
Detailsbinding site for residue 9SU A 1202
ChainResidue
ATYR1050
ATYR1060
APHE1061
AALA1062
ASER1068
ATYR1071
AGLY1074
AILE1075
AHOH1314
BGLU1138
AHIS1031
AGLY1032
APRO1034
APHE1035
AALA1049

site_idAC3
Number of Residues6
Detailsbinding site for residue PO4 A 1203
ChainResidue
AARG977
AHIS979
AARG980
AASP981
ALYS1067
BHOH1203

site_idAC4
Number of Residues7
Detailsbinding site for residue GOL A 1204
ChainResidue
ALYS996
ATYR1050
AMET1054
APHE1055
ATYR1060
ALYS1067
BGLU1138

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:O95271
ChainResidueDetails
ACYS1081
AHIS1084
ACYS1089
ACYS1092

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PDB entries from 2024-07-10

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