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6A5W

FXR-LBD with HNC143 and SRC1

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
A0032052molecular_functionbile acid binding
A0038183biological_processbile acid signaling pathway
C0003677molecular_functionDNA binding
C0004879molecular_functionnuclear receptor activity
C0006355biological_processregulation of DNA-templated transcription
C0032052molecular_functionbile acid binding
C0038183biological_processbile acid signaling pathway
Functional Information from PDB Data
site_idAC1
Number of Residues15
Detailsbinding site for residue 9R0 A 501
ChainResidue
ATHR270
AILE335
AHIS344
AHIS447
ATRP454
APHE461
ATRP469
AILE273
ALEU287
ATHR288
AMET290
AALA291
AMET328
APHE329
ASER332

site_idAC2
Number of Residues16
Detailsbinding site for residue 9R0 C 501
ChainResidue
CTHR270
CLEU287
CTHR288
CMET290
CALA291
CMET328
CPHE329
CSER332
CILE335
CHIS344
CLEU348
CTYR369
CHIS447
CTRP454
CPHE461
CTRP469

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsBinding site: {"evidences":[{"source":"PDB","id":"6HL1","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues2
DetailsModified residue: {"description":"Phosphothreonine; by PKC/PRKCZ","evidences":[{"source":"PubMed","id":"18668687","evidenceCode":"ECO:0000305"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues4
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO1)","evidences":[{"source":"PubMed","id":"23546875","evidenceCode":"ECO:0000305"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues8
DetailsMotif: {"description":"LXXLL motif 5"}
ChainResidueDetails

248335

PDB entries from 2026-01-28

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